DrugRepV Browse Page


DrugRepV browse page allows user to take a glance of the particular antiviral agent.Fields in the webpage is hylerlinked ot various external repositories like DrugBank, PubChem, Clinicaltrials.gov,and PubMed.User can explore the biological, Clinical, Chemical, and Structural details of every repurposed drug candidate.By clicking on the table header arrows, user can sort entries in ascending or descending order.


Total number of Records for Antiinfectives For Systemic Use are 889




DrugRepV_ID Antiviral Name
Drug type
Primary Indication
Secondary Indication
Strain
Pathways
Assay
Activity
Clinical Status
References
DrugRepV_0020Erythromycin
Antiinfectives For Systemic Use
Bacterial infections
Zika virus
GZ01, a recent Asian lineage
NA
Plaque assay
Increase (120 %)
Approved
29033372
DrugRepV_0046Sofosbuvir
Antiinfectives For Systemic Use
Hepatitis C virus | Acquired immunodeficiency syndrome
Zika virus
H/PF/2013
NA
Plaque assay
Decrease (50 %)
Approved
28912011
DrugRepV_0047Sofosbuvir
Antiinfectives For Systemic Use
Hepatitis C virus | Acquired immunodeficiency syndrome
Zika virus
H/PF/2013
NA
Cytopathic effect (CPE) assay
Decrease (50 %)
Approved
28912011
DrugRepV_0048Sofosbuvir
Antiinfectives For Systemic Use
Hepatitis C virus | Acquired immunodeficiency syndrome
Zika virus
ZIKVNL00013
NA
Plaque assay
Decrease (50 %)
Approved
28912011
DrugRepV_0049Sofosbuvir
Antiinfectives For Systemic Use
Hepatitis C virus | Acquired immunodeficiency syndrome
Zika virus
ZIKVNL00013
NA
Cytopathic effect (CPE) assay
Decrease (50 %)
Approved
28912011
DrugRepV_0050Sofosbuvir
Antiinfectives For Systemic Use
Hepatitis C virus | Acquired immunodeficiency syndrome
Zika virus
H/PF/2013
NA
Plaque assay
No significant effect (0 %)
Approved
28912011
DrugRepV_0051Sofosbuvir
Antiinfectives For Systemic Use
Hepatitis C virus | Acquired immunodeficiency syndrome
Zika virus
ZIKVNL00013
NA
Plaque assay
No significant effect (0 %)
Approved
28912011
DrugRepV_0052Sofosbuvir
Antiinfectives For Systemic Use
Hepatitis C virus | Acquired immunodeficiency syndrome
Zika virus
H/PF/2013
NA
Cytopathic effect (CPE) assay
No significant effect (0 %)
Approved
28912011
DrugRepV_0053Sofosbuvir
Antiinfectives For Systemic Use
Hepatitis C virus | Acquired immunodeficiency syndrome
Zika virus
ZIKVNL00013
NA
Cytopathic effect (CPE) assay
No significant effect (0 %)
Approved
28912011
DrugRepV_0054Sofosbuvir
Antiinfectives For Systemic Use
Hepatitis C virus | Acquired immunodeficiency syndrome
Zika virus
H/PF/2013
NA
Plaque assay
No significant effect (0 %)
Approved
28912011
DrugRepV_0055Sofosbuvir
Antiinfectives For Systemic Use
Hepatitis C virus | Acquired immunodeficiency syndrome
Zika virus
ZIKVNL00013
NA
Plaque assay
No significant effect (0 %)
Approved
28912011
DrugRepV_0202Azithromycin
Antiinfectives For Systemic Use
Microbial infections
Ebola virus
VLP
NA
Immunoflourescence assay
Decrease (50 %)
Approved
27890675
DrugRepV_0203Clarithromycin
Antiinfectives For Systemic Use
Microbial infections
Ebola virus
VLP
NA
Immunoflourescence assay
Decrease (50 %)
Approved
27890675
DrugRepV_0204Posaconazole
Antiinfectives For Systemic Use
Fungal infections (Aspergillus and Candida infections)
Ebola virus
VLP
NA
Immunoflourescence assay
Decrease (50 %)
Approved, Investigational, Vet approved
27890675
DrugRepV_0209Posaconazole
Antiinfectives For Systemic Use
Fungal infections (Aspergillus and Candida infections)
Ebola virus
EBOLA/Mayinga-eGFP
NA
Immunoflourescence assay
Decrease (50 %)
Approved, Investigational, Vet approved
27890675
DrugRepV_0211Clarithromycin
Antiinfectives For Systemic Use
Microbial infections
Ebola virus
EBOLA/Mayinga-eGFP
NA
Immunoflourescence assay
Decrease (50 %)
Approved
27890675
DrugRepV_0221Zidovudine
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome/AIDS
Ebola virus
ME718-1976/Yambuku-Ecran
NA
Real-time PCR
Increase (?3.12 ± 0.27 Ct)
Approved
27801778
DrugRepV_0222Zidovudine
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome/AIDS
Ebola virus
ME718-1976/Yambuku-Ecran
NA
Real-time PCR
Increase (?7.91 ± 2.67 Ct)
Approved
27801778
DrugRepV_0223Didanosine
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Ebola virus
ME718-1976/Yambuku-Ecran
NA
Real-time PCR
Increase (?0.43 ± 3.87 Ct)
Approved
27801778
DrugRepV_0224Didanosine
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Ebola virus
ME718-1976/Yambuku-Ecran
NA
Real-time PCR
Increase (?2.52 ± 1.27 Ct)
Approved
27801778
DrugRepV_0225Stavudine
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Ebola virus
ME718-1976/Yambuku-Ecran
NA
Real-time PCR
Increase (?2.87 ± 0.22 Ct)
Approved, Investigational
27801778
DrugRepV_0226Stavudine
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Ebola virus
ME718-1976/Yambuku-Ecran
NA
Real-time PCR
Increase (?3.93 ± 0.25 Ct)
Approved, Investigational
27801778
DrugRepV_0227Abacavir Sulfate
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Ebola virus
ME718-1976/Yambuku-Ecran
NA
Real-time PCR
Increase (?1.54 ± 3.26 Ct)
Approved
27801778
DrugRepV_0228Abacavir Sulfate
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Ebola virus
ME718-1976/Yambuku-Ecran
NA
Real-time PCR
Increase (?3.95 ± 2.69 Ct)
Approved
27801778
DrugRepV_0229Entecavir
Antiinfectives For Systemic Use
Hepatitis B virus
Ebola virus
ME718-1976/Yambuku-Ecran
NA
Real-time PCR
Increase (?3.08 ± 0.20 Ct)
Approved
27801778
DrugRepV_0230Entecavir
Antiinfectives For Systemic Use
Hepatitis B virus
Ebola virus
ME718-1976/Yambuku-Ecran
NA
Real-time PCR
Increase (?4.44 ± 1.11 Ct)
Approved
27801778
DrugRepV_0270Nalidixic Acid
Antiinfectives For Systemic Use
Bacterial infections
Influenza virus
A/New Jersey/15/2007
Pathway
Relative fluorescent unit
Decrease (50 %)
Approved, Investigational
26833677
DrugRepV_0271Nalidixic Acid
Antiinfectives For Systemic Use
Bacterial infections
Influenza virus
A/Netherlands/026/2008
Pathway
Relative fluorescent unit
Decrease (50 %)
Approved, Investigational
26833677
DrugRepV_0272Nalidixic Acid
Antiinfectives For Systemic Use
Bacterial infections
Influenza virus
A/Netherlands /049/2008
Pathway
Relative fluorescent unit
No significant effect (50 %)
Approved, Investigational
26833677
DrugRepV_0273Nalidixic Acid
Antiinfectives For Systemic Use
Bacterial infections
Influenza virus
A/Brisbane/59/2007
Pathway
Relative fluorescent unit
No significant effect (50 %)
Approved, Investigational
26833677
DrugRepV_0274Nalidixic Acid
Antiinfectives For Systemic Use
Bacterial infections
Influenza virus
A/New Jersey/15/2007
Pathway
Plaque assay
Decrease (10 %)
Approved, Investigational
26833677
DrugRepV_0275Nalidixic Acid
Antiinfectives For Systemic Use
Bacterial infections
Influenza virus
A/Brisbane/59/2007
Pathway
Plaque assay
No significant effect
Approved, Investigational
26833677
DrugRepV_0286Imipenem
Antiinfectives For Systemic Use
Bacterial infections
Influenza virus
A/New Jersey/15/2007
Pathway
Relative fluorescent unit
Decrease (50 %)
Approved
26833677
DrugRepV_0287Imipenem
Antiinfectives For Systemic Use
Bacterial infections
Influenza virus
A/Netherlands/026/2008
Pathway
Relative fluorescent unit
Decrease (50 %)
Approved
26833677
DrugRepV_0288Imipenem
Antiinfectives For Systemic Use
Bacterial infections
Influenza virus
A/Netherlands /049/2008
Pathway
Relative fluorescent unit
Decrease (50 %)
Approved
26833677
DrugRepV_0289Imipenem
Antiinfectives For Systemic Use
Bacterial infections
Influenza virus
A/Brisbane /56/2007
Pathway
Relative fluorescent unit
Decrease (50 %)
Approved
26833677
DrugRepV_0290Kaletra
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Middle East respiratory syndrome coronavirus
EMC/2012
NA
Real-time PCR
Decrease (1.06 Log10 Copies/GAPDH)
Approved, Investigational
26198719
DrugRepV_0291Kaletra
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Middle East respiratory syndrome coronavirus
EMC/2012
NA
Immunohistochemical assay
Decrease (>90 %)
Approved, Investigational
26198719
DrugRepV_0321Azithromycin
Antiinfectives For Systemic Use
Bacterial infections
Ebola virus
EBOV-eGFP
NA
Immunoflourescence assay
Decrease (50 %)
Approved
27622822
DrugRepV_0322Chlortetracycline
Antiinfectives For Systemic Use
Bacterial infections
Ebola virus
EBOV-eGFP
NA
Immunoflourescence assay
Decrease (50 %)
Approved
27622822
DrugRepV_0342Azithromycin
Antiinfectives For Systemic Use
Bacterial infections
Ebola virus
Ebola Zaire glycoprotein pseudotype vesicular stomatitis virus
NA
Renilla luciferase assay
Decrease (50 %)
Approved
27622822
DrugRepV_0343Chlortetracycline
Antiinfectives For Systemic Use
Bacterial infections
Ebola virus
Ebola Zaire glycoprotein pseudotype vesicular stomatitis virus
NA
Renilla luciferase assay
Decrease (50 %)
Approved
27622822
DrugRepV_0353Azithromycin
Antiinfectives For Systemic Use
Bacterial infections
Ebola virus
Ebola Zaire
NA
Survival assay
Increase
Approved
27622822
DrugRepV_0354Azithromycin
Antiinfectives For Systemic Use
Bacterial infections
Ebola virus
Ebola Zaire
NA
Survival assay
No significant effect
Approved
27622822
DrugRepV_0364Chlortetracycline
Antiinfectives For Systemic Use
Bacterial infections
Ebola virus
Ebola Zaire
NA
Survival assay
No significant effect
Approved
27622822
DrugRepV_0365Chlortetracycline
Antiinfectives For Systemic Use
Bacterial infections
Ebola virus
Ebola Zaire
NA
Survival assay
No significant effect
Approved
27622822
DrugRepV_0366Azithromycin
Antiinfectives For Systemic Use
Bacterial infections
Ebola virus
Ebola Mayinga
NA
Survival assay
No significant effect
Approved
27622822
DrugRepV_0374Cilastatin Sodium
Antiinfectives For Systemic Use
Bacterial infections
Ebola virus
eGFP-EBOV
NA
Fluorescence-based assay
Decrease (50 %)
Approved
26041706
DrugRepV_0384Flucytosine
Antiinfectives For Systemic Use
Fungal infections
Ebola virus
eGFP-EBOV
NA
Fluorescence-based assay
Decrease (50 %)
Approved, Investigational
26041706
DrugRepV_0431Efavirenz
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Ebola virus
eGFP-EBOV
NA
Fluorescence-based assay
Decrease (50 %)
Approved
26041706
DrugRepV_0445Teicoplanin
Antiinfectives For Systemic Use
Bacterial infections
Ebola virus
eGFP-EBOV
NA
Fluorescence-based assay
Decrease (50 %)
Approved
26041706
DrugRepV_0458Efavirenz
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Ebola virus
eGFP-EBOV
NA
Fluorescence-based assay
Decrease (50 %)
Approved
26041706
DrugRepV_0472Teicoplanin
Antiinfectives For Systemic Use
Bacterial infections
Ebola virus
eGFP-EBOV
NA
Fluorescence-based assay
Decrease (50 %)
Approved
26041706
DrugRepV_0487Efavirenz
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Ebola virus
EBOV-VLP
NA
Flow cytometry
Decrease (>90 %)
Approved
26041706
DrugRepV_0502Teicoplanin
Antiinfectives For Systemic Use
Bacterial infections
Ebola virus
EBOV-VLP
NA
Flow cytometry
Decrease (>90 %)
Approved
26041706
DrugRepV_0534Azithromycin
Antiinfectives For Systemic Use
Bacterial infections
Ebola virus
EBOVBlaVP40
NA
Fluorescence-based assay
Decrease (50 %)
Approved
26038505
DrugRepV_0537Clarithromycin
Antiinfectives For Systemic Use
Bacterial infections
Ebola virus
EBOVBlaVP40
NA
Fluorescence-based assay
Decrease (50 %)
Approved
26038505
DrugRepV_0556Spiramycin
Antiinfectives For Systemic Use
Bacterial infections
Ebola virus
EBOVBlaVP40
NA
Fluorescence-based assay
Decrease (50 %)
Approved
26038505
DrugRepV_0565Posaconazole
Antiinfectives For Systemic Use
Fungal infections (Aspergillus and Candida infections)
Ebola virus
EBOVBlaVP40
NA
Fluorescence-based assay
Decrease (50 %)
Approved, Investigational, Vet approved
26038505
DrugRepV_0580Minocycline
Antiinfectives For Systemic Use
Rocky Mountain spotted fever | Typhus fever and the typhus group | Q fever | Rickettsial pox | tick fevers caused by Rickettsiae | Upper respiratory tract infections caused by Streptococcus pneumoniae
Influenza virus
Anhui01
Pathway
Plaque assay
Decrease (1.3 Log10 copies)
Approved, Investigational
24496798
DrugRepV_0615Dirithromycin
Antiinfectives For Systemic Use
Bacterial infections
Lassa virus
GP derived Pseudovirus
NA
Luciferase reporter assay
No significant effect (0 %)
Approved
23577127
DrugRepV_0616Erythromycin
Antiinfectives For Systemic Use
Bacterial infections
Lassa virus
GP derived Pseudovirus
NA
Luciferase reporter assay
Decrease (60 %)
Approved
23577127
DrugRepV_0635Dirithromycin
Antiinfectives For Systemic Use
Bacterial infections
Lassa virus
Josiah
NA
Real-time PCR
No significant effect
Approved
23577127
DrugRepV_0636Erythromycin
Antiinfectives For Systemic Use
Bacterial infections
Lassa virus
Josiah
NA
Real-time PCR
No significant effect
Approved
23577127
DrugRepV_0654Dirithromycin
Antiinfectives For Systemic Use
Bacterial infections
Marburg virus
GP derived Pseudovirus
NA
Luciferase reporter assay
Decrease (91 %)
Approved
23577127
DrugRepV_0655Erythromycin
Antiinfectives For Systemic Use
Bacterial infections
Marburg virus
GP derived Pseudovirus
NA
Luciferase reporter assay
Decrease (98 %)
Approved
23577127
DrugRepV_0678Dirithromycin
Antiinfectives For Systemic Use
Bacterial infections
Ebola virus
GP derived Pseudovirus
NA
Luciferase reporter assay
Decrease (99 %)
Approved
23577127
DrugRepV_0679Erythromycin
Antiinfectives For Systemic Use
Bacterial infections
Ebola virus
GP derived Pseudovirus
NA
Luciferase reporter assay
Decrease (96 %)
Approved
23577127
DrugRepV_0700Dirithromycin
Antiinfectives For Systemic Use
Bacterial infections
Ebola virus
EBOLA-eGFP
NA
Fluorescence-based assay
No significant effect
Approved
23577127
DrugRepV_0701Erythromycin
Antiinfectives For Systemic Use
Bacterial infections
Ebola virus
EBOLA-eGFP
NA
Fluorescence-based assay
No significant effect
Approved
23577127
DrugRepV_0727Dirithromycin
Antiinfectives For Systemic Use
Bacterial infections
Ebola virus
ma-EBOV
NA
NA
No significant effect
Approved
23577127
DrugRepV_0728Erythromycin ethylsuccinate
Antiinfectives For Systemic Use
Bacterial infections
Ebola virus
ma-EBOV
NA
NA
No significant effect
Approved
23577127
DrugRepV_0760Clofazimine
Antiinfectives For Systemic Use
Lepromatous leprosy
Zika virus
MEX_I_7
NA
Fluorescence-based assay
Decrease (99.665 %)
Approved
27476412
DrugRepV_0782Daptomycin
Antiinfectives For Systemic Use
Bacterial infections
Zika virus
MEX_I_7
NA
Fluorescence-based assay
Decrease (89.915 %)
Approved
27476412
DrugRepV_0785Micafungin
Antiinfectives For Systemic Use
Fungal infections
Zika virus
MEX_I_7
NA
Fluorescence-based assay
Decrease (86.88 %)
Approved, Investigational
27476412
DrugRepV_0803Posaconazole
Antiinfectives For Systemic Use
Fungal infections (Aspergillus and Candida infections)
Zika virus
MEX_I_7
NA
Fluorescence-based assay
Decrease (61.34 %)
Approved, Investigational, Vet approved
27476412
DrugRepV_0839Isoniazid
Antiinfectives For Systemic Use
Tuberculosis
Zika virus
MEX_I_7
NA
Fluorescence-based assay
Decrease (60.29 %)
Approved, Investigational
27476412
DrugRepV_0843Penicillin G Potassium
Antiinfectives For Systemic Use
Septicemia | Meningitis | Pericarditis | Endocarditis | Pneumonia
Zika virus
MEX_I_7
NA
Fluorescence-based assay
Decrease (52.15 %)
Approved
27476412
DrugRepV_0846Cefuroxime Axetil
Antiinfectives For Systemic Use
Bacterial infections
Zika virus
MEX_I_7
NA
Fluorescence-based assay
Decrease (55.5 %)
Approved
27476412
DrugRepV_0852Linezolid
Antiinfectives For Systemic Use
Bacterial infections
Zika virus
MEX_I_7
NA
Fluorescence-based assay
Decrease (60.395 %)
Approved, Investigational
27476412
DrugRepV_0856Lincomycin Hydrochloride
Antiinfectives For Systemic Use
Bacterial infections
Zika virus
MEX_I_7
NA
Fluorescence-based assay
Decrease (58.795 %)
Approved, Vet approved
27476412
DrugRepV_0859Nelfinavir Mesylate
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Zika virus
MEX_I_7
NA
Fluorescence-based assay
Decrease (60.53 %)
Approved
27476412
DrugRepV_0870Erythromycin
Antiinfectives For Systemic Use
Bacterial infections
Zika virus
MEX_I_7
NA
Fluorescence-based assay
Decrease (55.1 %)
Approved
27476412
DrugRepV_0876Norfloxacin
Antiinfectives For Systemic Use
Urinary tract infection
Zika virus
MEX_I_7
NA
Fluorescence-based assay
Decrease (57.51 %)
Approved
27476412
DrugRepV_0878Amphotericin B
Antiinfectives For Systemic Use
Fungal infections
Zika virus
MEX_I_7
NA
Fluorescence-based assay
Decrease (54.04 %)
Approved
27476412
DrugRepV_0886Ketoconazole
Antiinfectives For Systemic Use
Fungal infections
Zika virus
MEX_I_7
NA
Fluorescence-based assay
Decrease (60.415 %)
Approved, Investigational
27476412
DrugRepV_0888Ceftibuten
Antiinfectives For Systemic Use
Bacterial infections
Zika virus
MEX_I_7
NA
Fluorescence-based assay
Decrease (53.895 %)
Approved
27476412
DrugRepV_0901Efavirenz
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Zika virus
MEX_I_7
NA
Fluorescence-based assay
Decrease (57.92 %)
Approved
27476412
DrugRepV_0907Ofloxacin
Antiinfectives For Systemic Use
Respiratory tract infections | Kidney infection | Skin infection
Zika virus
MEX_I_7
NA
Fluorescence-based assay
Decrease (55.695 %)
Approved
27476412
DrugRepV_0909Penciclovir
Antiinfectives For Systemic Use
Recurrent cold sores on the lips and face from Herpesvirus invections
Zika virus
MEX_I_7
NA
Fluorescence-based assay
Decrease (55.495 %)
Approved
27476412
DrugRepV_0923Amikacin Disulfate
Antiinfectives For Systemic Use
Bacterial infections
Zika virus
MEX_I_7
NA
Fluorescence-based assay
Decrease (52.975 %)
Approved
27476412
DrugRepV_0924Ciprofloxacin
Antiinfectives For Systemic Use
Bacterial infections
Zika virus
MEX_I_7
NA
Fluorescence-based assay
Decrease (55.87 %)
Approved
27476412
DrugRepV_0926Spectinomycin Hydrochloride Pentahydrate
Antiinfectives For Systemic Use
Bacterial infections (Gonorrheal urethritis and proctitis)
Zika virus
MEX_I_7
NA
Fluorescence-based assay
Decrease (55.825 %)
Approved, Investigational, Vet approved
27476412
DrugRepV_0937Penicillin V Potassium
Antiinfectives For Systemic Use
Mild to moderately severe infections due to penicillin G­-sensitive microorganisms
Zika virus
MEX_I_7
NA
Fluorescence-based assay
Decrease (52.165 %)
Approved
27476412
DrugRepV_0938Ceftriaxone Sodium
Antiinfectives For Systemic Use
Bacterial infections
Zika virus
MEX_I_7
NA
Fluorescence-based assay
Decrease (55.04 %)
Approved
27476412
DrugRepV_0963Zanamivir
Antiinfectives For Systemic Use
Influenza virus
Zika virus
MEX_I_7
NA
Fluorescence-based assay
Decrease (47.235 %)
Approved
27476412
DrugRepV_0968Ethionamide
Antiinfectives For Systemic Use
Tuberculosis
Zika virus
MEX_I_7
NA
Fluorescence-based assay
Decrease (52.99 %)
Approved
27476412
DrugRepV_0974Oxacillin Sodium salt Monohydrate
Antiinfectives For Systemic Use
Staphylococci infections
Zika virus
MEX_I_7
NA
Fluorescence-based assay
Decrease (54.525 %)
Approved, Investigational
27476412
DrugRepV_0982Cefixime
Antiinfectives For Systemic Use
Bacterial infections
Zika virus
MEX_I_7
NA
Fluorescence-based assay
Decrease (48.925 %)
Approved
27476412
DrugRepV_0986Pyrazinamide
Antiinfectives For Systemic Use
Tuberculosis
Zika virus
MEX_I_7
NA
Fluorescence-based assay
Decrease (50.975 %)
Approved, Investigational
27476412
DrugRepV_1001Delavirdine Mesylate
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Zika virus
MEX_I_7
NA
Fluorescence-based assay
Decrease (54.035 %)
Approved
27476412
DrugRepV_1012Cefaclor
Antiinfectives For Systemic Use
Bacterial infections
Zika virus
MEX_I_7
NA
Fluorescence-based assay
Decrease (50.11 %)
Approved
27476412
DrugRepV_1015Chloramphenicol
Antiinfectives For Systemic Use
Bacterial infections
Zika virus
MEX_I_7
NA
Fluorescence-based assay
Decrease (54.08 %)
Approved
27476412
DrugRepV_1020Cidofovir
Antiinfectives For Systemic Use
Cytomegalovirus infection
Zika virus
MEX_I_7
NA
Fluorescence-based assay
Decrease (53.06 %)
Approved
27476412
DrugRepV_1021Levofloxacin Hydrochloride
Antiinfectives For Systemic Use
Bacterial infections (Conjunctivitis)
Zika virus
MEX_I_7
NA
Fluorescence-based assay
Decrease (51.885 %)
Approved
27476412
DrugRepV_1022Demeclocycline Hydrochloride
Antiinfectives For Systemic Use
Bacterial infections
Zika virus
MEX_I_7
NA
Fluorescence-based assay
Decrease (50.41 %)
Approved
27476412
DrugRepV_1026Cefuroxime Sodium
Antiinfectives For Systemic Use
Bacterial infections
Zika virus
MEX_I_7
NA
Fluorescence-based assay
Decrease (52.005 %)
Approved
27476412
DrugRepV_1029Ethambutol Dihydrochloride
Antiinfectives For Systemic Use
Bacterial infections
Zika virus
MEX_I_7
NA
Fluorescence-based assay
Decrease (49.32 %)
Approved
27476412
DrugRepV_1035Doxycycline Monohydrate
Antiinfectives For Systemic Use
Bacterial infections
Zika virus
MEX_I_7
NA
Fluorescence-based assay
Decrease (52.935 %)
Approved
27476412
DrugRepV_1043Voriconazole
Antiinfectives For Systemic Use
Fungal infections
Zika virus
MEX_I_7
NA
Fluorescence-based assay
Decrease (52.235 %)
Approved
27476412
DrugRepV_1045Dapsone
Antiinfectives For Systemic Use
Leprosy and dermatitis herpetiformis
Zika virus
MEX_I_7
NA
Fluorescence-based assay
Decrease (48.585 %)
Approved
27476412
DrugRepV_1053Bacitracin
Antiinfectives For Systemic Use
Bacterial infections
Zika virus
MEX_I_7
NA
Fluorescence-based assay
Decrease (47.205 %)
Approved
27476412
DrugRepV_1055Ceftizoxim Sodium
Antiinfectives For Systemic Use
Bacterial infections
Zika virus
MEX_I_7
NA
Fluorescence-based assay
Decrease (52.58 %)
Approved
27476412
DrugRepV_1075Cefotaxime Acid
Antiinfectives For Systemic Use
Bacterial infections
Zika virus
MEX_I_7
NA
Fluorescence-based assay
Decrease (54.85 %)
Approved
27476412
DrugRepV_1076Lopinavir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Zika virus
MEX_I_7
NA
Fluorescence-based assay
Decrease (55 %)
Approved
27476412
DrugRepV_1078Clindamycin Hydrochloride
Antiinfectives For Systemic Use
Bacterial infections
Zika virus
MEX_I_7
NA
Fluorescence-based assay
Decrease (51.415 %)
Approved
27476412
DrugRepV_1084Gemifloxacin
Antiinfectives For Systemic Use
Bacterial infections (Chronic bronchitis and mild-to-moderate pneumonia)
Zika virus
MEX_I_7
NA
Fluorescence-based assay
Decrease (51.92 %)
Approved, Investigational
27476412
DrugRepV_1085Adefovir dipivoxil
Antiinfectives For Systemic Use
Hepatitis B virus
Zika virus
MEX_I_7
NA
Fluorescence-based assay
Decrease (52.3 %)
Approved
27476412
DrugRepV_1090Cefprozil
Antiinfectives For Systemic Use
Bacterial infections
Zika virus
MEX_I_7
NA
Fluorescence-based assay
Decrease (46.765 %)
Approved
27476412
DrugRepV_1095Emtricitabine
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Zika virus
MEX_I_7
NA
Fluorescence-based assay
Decrease (51.065 %)
Approved
27476412
DrugRepV_1096Cefdinir
Antiinfectives For Systemic Use
Bacterial infections
Zika virus
MEX_I_7
NA
Fluorescence-based assay
Decrease (47.845 %)
Approved
27476412
DrugRepV_1103Cycloserine
Antiinfectives For Systemic Use
Tuberculosis
Zika virus
MEX_I_7
NA
Fluorescence-based assay
Decrease (47.77 %)
Approved
27476412
DrugRepV_1109Tenofovir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Zika virus
MEX_I_7
NA
Fluorescence-based assay
Decrease (44.855 %)
Approved, Investigational
27476412
DrugRepV_1111Moxifloxacin Hydrochloride
Antiinfectives For Systemic Use
Sinusitis | Pneumonia | Chronic bronchitis
Zika virus
MEX_I_7
NA
Fluorescence-based assay
Decrease (53.71 %)
Approved, Investigational
27476412
DrugRepV_1113Oxytetracycline Hydrochloride
Antiinfectives For Systemic Use
Bacterial infections
Zika virus
MEX_I_7
NA
Fluorescence-based assay
Decrease (46.71 %)
Approved, Investigational, Vet approved
27476412
DrugRepV_1116Valganciclovir Hydrochloride
Antiinfectives For Systemic Use
Herpes simplex and Zoster virus
Zika virus
MEX_I_7
NA
Fluorescence-based assay
Decrease (49.32 %)
Approved
27476412
DrugRepV_11184-Aminosalicylic Acid
Antiinfectives For Systemic Use
Tuberculosis
Zika virus
MEX_I_7
NA
Fluorescence-based assay
Decrease (51.44 %)
Approved
27476412
DrugRepV_1131Methenamine Hippurate
Antiinfectives For Systemic Use
Urinary tract infection
Zika virus
MEX_I_7
NA
Fluorescence-based assay
Decrease (52.645 %)
Approved, Vet approved
27476412
DrugRepV_1132Cloxacillin Sodium
Antiinfectives For Systemic Use
Bacterial infections
Zika virus
MEX_I_7
NA
Fluorescence-based assay
Decrease (49.82 %)
Approved
27476412
DrugRepV_1148Piperacillin
Antiinfectives For Systemic Use
Polymicrobial infections
Zika virus
MEX_I_7
NA
Fluorescence-based assay
Decrease (47.9 %)
Approved
27476412
DrugRepV_1151Famciclovir
Antiinfectives For Systemic Use
Herpes simplex virus | Zoster virus
Zika virus
MEX_I_7
NA
Fluorescence-based assay
Decrease (47.62 %)
Approved, Investigational
27476412
DrugRepV_1157Amoxicillin
Antiinfectives For Systemic Use
Bacterial infections
Zika virus
MEX_I_7
NA
Fluorescence-based assay
Decrease (49.335 %)
Approved
27476412
DrugRepV_1163Sulfanilamide
Antiinfectives For Systemic Use
Vulvovaginitis
Zika virus
MEX_I_7
NA
Fluorescence-based assay
Decrease (47.175 %)
Approved
27476412
DrugRepV_1165Rifampin
Antiinfectives For Systemic Use
Tuberculosis and Tuberculosis-related mycobacterial infections
Zika virus
MEX_I_7
NA
Fluorescence-based assay
Decrease (52.505 %)
Approved
27476412
DrugRepV_1167Cefepime Hydrochloride Hydrate
Antiinfectives For Systemic Use
Bacterial infections
Zika virus
MEX_I_7
NA
Fluorescence-based assay
Decrease (52.89 %)
Approved
27476412
DrugRepV_1177Doripenem
Antiinfectives For Systemic Use
Intra-abdominal infections and complicated urinary tract infections
Zika virus
MEX_I_7
NA
Fluorescence-based assay
Decrease (47.47 %)
Approved
27476412
DrugRepV_1187Cefadroxil
Antiinfectives For Systemic Use
Bacterial infections
Zika virus
MEX_I_7
NA
Fluorescence-based assay
Decrease (48.15 %)
Approved
27476412
DrugRepV_1189Raltegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Zika virus
MEX_I_7
NA
Fluorescence-based assay
Decrease (49.03 %)
Approved
27476412
DrugRepV_1191Dicloxacillin Sodium Salt Monohydrate
Antiinfectives For Systemic Use
Bacterial infections
Zika virus
MEX_I_7
NA
Fluorescence-based assay
Decrease (46.765 %)
Approved
27476412
DrugRepV_1196Ganciclovir
Antiinfectives For Systemic Use
Cytomegalovirus infection
Zika virus
MEX_I_7
NA
Fluorescence-based assay
Decrease (49.48 %)
Approved, Investigational
27476412
DrugRepV_1209Maraviroc
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Zika virus
MEX_I_7
NA
Fluorescence-based assay
Decrease (48.18 %)
Approved, Investigational
27476412
DrugRepV_1212Zalcitabine
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome/AIDS
Zika virus
MEX_I_7
NA
Fluorescence-based assay
Decrease (49.06 %)
Approved
27476412
DrugRepV_1216Kanamycin Sulfate
Antiinfectives For Systemic Use
Bacterial infections
Zika virus
MEX_I_7
NA
Fluorescence-based assay
Decrease (46.43 %)
Approved, Investigational, Vet approved
27476412
DrugRepV_1225Nevirapine
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Zika virus
MEX_I_7
NA
Fluorescence-based assay
Decrease (47.07 %)
Approved
27476412
DrugRepV_1227Darunavir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Zika virus
MEX_I_7
NA
Fluorescence-based assay
Decrease (44.605 %)
Approved
27476412
DrugRepV_1234Cefotetan Disodium
Antiinfectives For Systemic Use
Bacterial infections
Zika virus
MEX_I_7
NA
Fluorescence-based assay
Decrease (47.645 %)
Approved
27476412
DrugRepV_1235Aztreonam
Antiinfectives For Systemic Use
Bacterial infections
Zika virus
MEX_I_7
NA
Fluorescence-based assay
Decrease (46.05 %)
Approved
27476412
DrugRepV_1238Flucytosine
Antiinfectives For Systemic Use
Fungal infections
Zika virus
MEX_I_7
NA
Fluorescence-based assay
Decrease (48.75 %)
Approved, Investigational
27476412
DrugRepV_1247Minocycline
Antiinfectives For Systemic Use
Rocky Mountain spotted fever | Typhus fever and the typhus group | Q fever | Rickettsial pox | tick fevers caused by Rickettsiae | Upper respiratory tract infections caused by Streptococcus pneumoniae
Zika virus
MEX_I_7
NA
Fluorescence-based assay
Decrease (46.405 %)
Approved, Investigational
27476412
DrugRepV_1261Ritonavir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Zika virus
MEX_I_7
NA
Fluorescence-based assay
Decrease (40.915 %)
Approved, Investigational
27476412
DrugRepV_1262Cefditoren Pivoxil
Antiinfectives For Systemic Use
Bacterial infections
Zika virus
MEX_I_7
NA
Fluorescence-based assay
Decrease (46.4 %)
Approved
27476412
DrugRepV_1264Cefpodoxime Proxetil
Antiinfectives For Systemic Use
Bacterial infections
Zika virus
MEX_I_7
NA
Fluorescence-based assay
Decrease (46.81 %)
Approved
27476412
DrugRepV_1271Meropenem
Antiinfectives For Systemic Use
Bacterial infections (Skin infection)
Zika virus
MEX_I_7
NA
Fluorescence-based assay
Decrease (48.025 %)
Approved, Investigational
27476412
DrugRepV_1274Lamivudine
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome | Hepatitis B virus
Zika virus
MEX_I_7
NA
Fluorescence-based assay
Decrease (45.2 %)
Approved, Investigational
27476412
DrugRepV_1276Tigecycline
Antiinfectives For Systemic Use
Complicated skin and skin structure infections
Zika virus
MEX_I_7
NA
Fluorescence-based assay
Decrease (46.4 %)
Approved
27476412
DrugRepV_1281Clarithromycin
Antiinfectives For Systemic Use
Microbial infections
Zika virus
MEX_I_7
NA
Fluorescence-based assay
Decrease (49.09 %)
Approved
27476412
DrugRepV_1282Fosfomycin Calcium
Antiinfectives For Systemic Use
Bacterial infections
Zika virus
MEX_I_7
NA
Fluorescence-based assay
Decrease (45.385 %)
Approved
27476412
DrugRepV_1288Trimethoprim
Antiinfectives For Systemic Use
Urinary tract infections | Uncomplicated pyelonephritis (with sulfamethoxazole) | Mild acute prostatitis
Zika virus
MEX_I_7
NA
Fluorescence-based assay
Decrease (49.69 %)
Approved
27476412
DrugRepV_1295Cilastatin Sodium
Antiinfectives For Systemic Use
Bacterial infections
Zika virus
MEX_I_7
NA
Fluorescence-based assay
Decrease (49.065 %)
Approved
27476412
DrugRepV_1302Stavudine
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Zika virus
MEX_I_7
NA
Fluorescence-based assay
Decrease (45.29 %)
Approved, Investigational
27476412
DrugRepV_1307Neomycin Sulfate
Antiinfectives For Systemic Use
Bacterial infections
Zika virus
MEX_I_7
NA
Fluorescence-based assay
Decrease (47.33 %)
Approved
27476412
DrugRepV_1309Nafcillin Sodium
Antiinfectives For Systemic Use
Bacterial infections
Zika virus
MEX_I_7
NA
Fluorescence-based assay
Decrease (42.57 %)
Approved, Investigational
27476412
DrugRepV_1310Capreomycin Disulfate
Antiinfectives For Systemic Use
Tuberculosis
Zika virus
MEX_I_7
NA
Fluorescence-based assay
Decrease (46.425 %)
Approved
27476412
DrugRepV_1321Sulfamethoxazole
Antiinfectives For Systemic Use
Bacterial infections (Bronchitis, prostatitis and urinary tract infections)
Zika virus
MEX_I_7
NA
Fluorescence-based assay
Decrease (43.87 %)
Approved
27476412
DrugRepV_1325Tetracycline
Antiinfectives For Systemic Use
Bacterial infections (Rocky Mountain spotted fever | Typhus fever | Tick fevers | Q fever | Rickettsialpox | Brill-Zinsser disease)
Zika virus
MEX_I_7
NA
Fluorescence-based assay
Decrease (49.51 %)
Approved
27476412
DrugRepV_1326Sulfadiazine
Antiinfectives For Systemic Use
Rheumatic fever | Meningococcal meningitis
Zika virus
MEX_I_7
NA
Fluorescence-based assay
Decrease (48.975 %)
Approved, Investigational, Vet approved
27476412
DrugRepV_1340Itraconazole
Antiinfectives For Systemic Use
Fungal infections (Pulmonary and extrapulmonary blastomycosis, Histoplasmosis, Aspergillosis, and Onychomycosis)
Zika virus
MEX_I_7
NA
Fluorescence-based assay
Decrease (47.185 %)
Approved, Investigational
27476412
DrugRepV_1352Gatifloxacin
Antiinfectives For Systemic Use
Bacterial infections (Bronchitis, sinusitis, Community-acquired pneumonia, and Skin infections)
Zika virus
MEX_I_7
NA
Fluorescence-based assay
Decrease (45.98 %)
Approved, Investigational
27476412
DrugRepV_1362Zidovudine
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome/AIDS
Zika virus
MEX_I_7
NA
Fluorescence-based assay
Decrease (46.965 %)
Approved
27476412
DrugRepV_1364Telbivudine
Antiinfectives For Systemic Use
Hepatitis B virus
Zika virus
MEX_I_7
NA
Fluorescence-based assay
Decrease (44.765 %)
Approved
27476412
DrugRepV_1369Fluconazole
Antiinfectives For Systemic Use
Fungal infections
Zika virus
MEX_I_7
NA
Fluorescence-based assay
Decrease (40.98 %)
Approved, Investigational
27476412
DrugRepV_1371Azithromycin
Antiinfectives For Systemic Use
Microbial infections
Zika virus
MEX_I_7
NA
Fluorescence-based assay
Decrease (44.07 %)
Approved
27476412
DrugRepV_1380Ampicillin Trihydrate
Antiinfectives For Systemic Use
Bacterial infections
Zika virus
MEX_I_7
NA
Fluorescence-based assay
Decrease (46.895 %)
Approved
27476412
DrugRepV_1382Foscarnet Sodium
Antiinfectives For Systemic Use
Cytomegalovirus retinitis | Herpesviruses | Acquired immunodeficiency syndrome
Zika virus
MEX_I_7
NA
Fluorescence-based assay
Decrease (42.945 %)
Approved
27476412
DrugRepV_1391Nitrofurantoin
Antiinfectives For Systemic Use
Urinary tract infection
Zika virus
MEX_I_7
NA
Fluorescence-based assay
Decrease (45.26 %)
Approved
27476412
DrugRepV_1392Abacavir Sulfate
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Zika virus
MEX_I_7
NA
Fluorescence-based assay
Decrease (45.76 %)
Approved
27476412
DrugRepV_1416Rifapentine
Antiinfectives For Systemic Use
Tuberculosis
Zika virus
MEX_I_7
NA
Fluorescence-based assay
Decrease (41.79 %)
Approved, Investigational
27476412
DrugRepV_1433Idoxuridine
Antiinfectives For Systemic Use
Keratoconjunctivitis and Keratitis caused by herpes simplex virus
Zika virus
MEX_I_7
NA
Fluorescence-based assay
Decrease (42.78 %)
Approved, Investigational
27476412
DrugRepV_1444Ribavirin
Antiinfectives For Systemic Use
Hepatitis C virus
Zika virus
MEX_I_7
NA
Fluorescence-based assay
Decrease (43.21 %)
Approved
27476412
DrugRepV_1450Valacyclovir Hydrochloride
Antiinfectives For Systemic Use
Herpes simplex and Zoster virus
Zika virus
MEX_I_7
NA
Fluorescence-based assay
Decrease (44.35 %)
Approved
27476412
DrugRepV_1454Didanosine
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Zika virus
MEX_I_7
NA
Fluorescence-based assay
Decrease (40.17 %)
Approved
27476412
DrugRepV_1457Imipenem
Antiinfectives For Systemic Use
Bacterial infections
Zika virus
MEX_I_7
NA
Fluorescence-based assay
Decrease (42.8 %)
Approved
27476412
DrugRepV_1460Indinavir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Zika virus
MEX_I_7
NA
Fluorescence-based assay
Decrease (42.985 %)
Approved
27476412
DrugRepV_1478Atazanavir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Zika virus
MEX_I_7
NA
Fluorescence-based assay
Decrease (38.68 %)
Approved
27476412
DrugRepV_1482Rifabutin
Antiinfectives For Systemic Use
Mycobacterium avium complex (MAC) disease in patients with advanced Acquired immunodeficiency syndrome infection
Zika virus
MEX_I_7
NA
Fluorescence-based assay
Decrease (35.56 %)
Approved, Investigational
27476412
DrugRepV_1486Oseltamivir Phosphate
Antiinfectives For Systemic Use
Influenza A/B virus
Zika virus
MEX_I_7
NA
Fluorescence-based assay
Decrease (44.305 %)
Approved
27476412
DrugRepV_1501Rimantadine Hydrochloride
Antiinfectives For Systemic Use
Influenza A virus
Zika virus
MEX_I_7
NA
Fluorescence-based assay
Decrease (39.755 %)
Approved, Investigational
27476412
DrugRepV_1516Saquinavir Mesylate
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Zika virus
MEX_I_7
NA
Fluorescence-based assay
Decrease (32.635 %)
Approved, Investigational
27476412
DrugRepV_1517Telithromycin
Antiinfectives For Systemic Use
Pneumococcal infection | Acute sinusitis | Acute bacterial tonsillitis | Acute bronchitis and bronchiolitis | Lower respiratory tract infection and lobar (pneumococcal) pneumonia
Zika virus
MEX_I_7
NA
Fluorescence-based assay
Decrease (31.37 %)
Approved
27476412
DrugRepV_1522Streptomycin Sulfate
Antiinfectives For Systemic Use
Tuberculosis | Tularemia | Plague | Brucellosis | Endocarditis
Zika virus
MEX_I_7
NA
Fluorescence-based assay
Decrease (28.56 %)
Approved, Vet approved
27476412
DrugRepV_1530Clindamycin Palmitate Hydrochloride
Antiinfectives For Systemic Use
Bacterial infections
Zika virus
MEX_I_7
NA
Fluorescence-based assay
Decrease (22.29 %)
Approved
27476412
DrugRepV_1534Daptomycin
Antiinfectives For Systemic Use
Bacterial infections
Zika virus
MEX_I_7
NA
Flow cytometry
Decrease (50 %)
Approved
27476412
DrugRepV_1541Daptomycin
Antiinfectives For Systemic Use
Bacterial infections
Zika virus
MEX_I_7
NA
Flow cytometry
No significant effect (50 %)
Approved
27476412
DrugRepV_1545Daptomycin
Antiinfectives For Systemic Use
Bacterial infections
Zika virus
MEX_I_7
NA
Flow cytometry
Increase (120 %)
Approved
27476412
DrugRepV_1550Daptomycin
Antiinfectives For Systemic Use
Bacterial infections
Zika virus
DAK_41525
NA
Flow cytometry
No significant effect
Approved
27476412
DrugRepV_1557Daptomycin
Antiinfectives For Systemic Use
Bacterial infections
Zika virus
MEX_I_7
NA
Fluorescence-based assay
Decrease (50 %)
Approved
27476412
DrugRepV_1576Itraconazole
Antiinfectives For Systemic Use
Fungal infections (Pulmonary and extrapulmonary blastomycosis, Histoplasmosis, Aspergillosis, and Onychomycosis)
Rift Valley fever virus
MP12-Luc
NA
Luciferase reporter assay
Decrease (74 %)
Approved, Investigational
26217313
DrugRepV_1592Ribavirin
Antiinfectives For Systemic Use
Hepatitis C virus
Rift Valley fever virus
rMP12
NA
Plaque assay
Decrease (4 Logs reduction)
Approved
26217313
DrugRepV_1594Ribavirin
Antiinfectives For Systemic Use
Hepatitis C virus
Rift Valley fever virus
rMP12
NA
Plaque assay
Decrease (4.5 Logs reduction)
Approved
26217313
DrugRepV_1596Ribavirin
Antiinfectives For Systemic Use
Hepatitis C virus
Rift Valley fever virus
rMP12
NA
Plaque assay
Decrease (1 Logs reduction)
Approved
26217313
DrugRepV_1598Ribavirin
Antiinfectives For Systemic Use
Hepatitis C virus
Rift Valley fever virus
rMP12
NA
Plaque assay
Decrease (3 Logs reduction)
Approved
26217313
DrugRepV_1600Ribavirin
Antiinfectives For Systemic Use
Hepatitis C virus
Rift Valley fever virus
rMP12
NA
Plaque assay
Decrease (4 Logs reduction)
Approved
26217313
DrugRepV_1602Ribavirin
Antiinfectives For Systemic Use
Hepatitis C virus
Rift Valley fever virus
rMP12
NA
Plaque assay
Decrease (6 Logs reduction)
Approved
26217313
DrugRepV_1604Ribavirin
Antiinfectives For Systemic Use
Hepatitis C virus
Rift Valley fever virus
rMP12
NA
Plaque assay
Decrease (2 Logs reduction)
Approved
26217313
DrugRepV_1606Ribavirin
Antiinfectives For Systemic Use
Hepatitis C virus
Rift Valley fever virus
rMP12
NA
Plaque assay
Decrease (5 Logs reduction)
Approved
26217313
DrugRepV_1608Ribavirin
Antiinfectives For Systemic Use
Hepatitis C virus
Rift Valley fever virus
rMP12
NA
Plaque assay
Decrease (100 %)
Approved
26217313
DrugRepV_1622Minocycline
Antiinfectives For Systemic Use
Rocky Mountain spotted fever | Typhus fever and the typhus group | Q fever | Rickettsial pox | tick fevers caused by Rickettsiae | Upper respiratory tract infections caused by Streptococcus pneumoniae
Influenza virus
A/Anhui/01/2013
Pathway
Transcriptomic response-DEG
Decrease
Approved, Investigational
24991006
DrugRepV_1930Nelfinavir Mesylate
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Zika virus
H/PF/2013
NA
Plaque assay
Decrease (2 Logs)
Approved
28814523
DrugRepV_1935Nelfinavir Mesylate
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Zika virus
H/PF/2013
NA
Real-time PCR
Decrease (0 %)
Approved
28814523
DrugRepV_1940Nelfinavir Mesylate
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Zika virus
H/PF/2013
NA
Immunoflourescence assay
Decrease
Approved
28814523
DrugRepV_2015Teicoplanin
Antiinfectives For Systemic Use
Bacterial infections
Ebola virus
Zaire strain-pEBOV
NA
Firefly luciferase assay
Decrease (50 %)
Approved
26585243
DrugRepV_2030Teicoplanin
Antiinfectives For Systemic Use
Bacterial infections
Ebola virus
Zaire strain-pEBOV
NA
Firefly luciferase assay
Decrease (90 %)
Approved
26585243
DrugRepV_2031Teicoplanin
Antiinfectives For Systemic Use
Bacterial infections
Ebola virus
Zaire strain-pEBOV
NA
Firefly luciferase assay
Decrease (50 %)
Approved
26585243
DrugRepV_2032Teicoplanin
Antiinfectives For Systemic Use
Bacterial infections
Ebola virus
Zaire strain-pEBOV
NA
Firefly luciferase assay
Decrease (87.5 %)
Approved
26585243
DrugRepV_2033Teicoplanin
Antiinfectives For Systemic Use
Bacterial infections
Ebola virus
Zaire strain-pEBOV
NA
Firefly luciferase assay
Decrease (95 %)
Approved
26585243
DrugRepV_2034Teicoplanin
Antiinfectives For Systemic Use
Bacterial infections
Ebola virus
Zaire strain-pEBOV
NA
Firefly luciferase assay
No significant effect (0 %)
Approved
26585243
DrugRepV_2038Lopinavir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Middle East respiratory syndrome coronavirus
EMC/2012
NA
Cell viability assay
Decrease (50 %)
Approved
24841269
DrugRepV_2042Lopinavir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Severe acute respiratory syndrome coronavirus
NA
NA
Cell viability assay
Decrease (50 %)
Approved
24841269
DrugRepV_2046Lopinavir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Severe acute respiratory syndrome coronavirus
229E-GFP
NA
Cell viability assay
Decrease (50 %)
Approved
24841269
DrugRepV_2052Rifabutin
Antiinfectives For Systemic Use
Mycobacterium avium complex (MAC) disease in patients with advanced Acquired immunodeficiency syndrome infection
Middle East respiratory syndrome coronavirus
EMC/2012
NA
Cell viability assay
No significant decrease (10 %)
Approved, Investigational
24841269
DrugRepV_2053Rifapentine
Antiinfectives For Systemic Use
Tuberculosis
Middle East respiratory syndrome coronavirus
EMC/2012
NA
Cell viability assay
Decrease (50 %)
Approved, Investigational
24841269
DrugRepV_2113Sofosbuvir
Antiinfectives For Systemic Use
Hepatitis C virus | Acquired immunodeficiency syndrome
Zika virus
PRVABC-59
NA
Plaque assay
Decrease (50 %)
Approved
27902933
DrugRepV_2114Sofosbuvir
Antiinfectives For Systemic Use
Hepatitis C virus | Acquired immunodeficiency syndrome
Zika virus
PRVABC-59
NA
Plaque assay
Decrease (50 %)
Approved
27902933
DrugRepV_2115Sofosbuvir
Antiinfectives For Systemic Use
Hepatitis C virus | Acquired immunodeficiency syndrome
Zika virus
Paraiba
NA
Plaque assay
Decrease (50 %)
Approved
27902933
DrugRepV_2116Sofosbuvir
Antiinfectives For Systemic Use
Hepatitis C virus | Acquired immunodeficiency syndrome
Zika virus
Paraiba
NA
Plaque assay
Decrease (50 %)
Approved
27902933
DrugRepV_2117Sofosbuvir
Antiinfectives For Systemic Use
Hepatitis C virus | Acquired immunodeficiency syndrome
Zika virus
Dakar
NA
Plaque assay
Decrease (50 %)
Approved
27902933
DrugRepV_2118Sofosbuvir
Antiinfectives For Systemic Use
Hepatitis C virus | Acquired immunodeficiency syndrome
Zika virus
Dakar
NA
Plaque assay
Decrease (50 %)
Approved
27902933
DrugRepV_2119Sofosbuvir
Antiinfectives For Systemic Use
Hepatitis C virus | Acquired immunodeficiency syndrome
Zika virus
PRVABC-59
NA
Real-time PCR
Decrease (>1 Log10 (GE/ml))
Approved
27902933
DrugRepV_2120Sofosbuvir
Antiinfectives For Systemic Use
Hepatitis C virus | Acquired immunodeficiency syndrome
Zika virus
PRVABC-59
NA
Real-time PCR
Decrease (2 Log10 (GE/ml))
Approved
27902933
DrugRepV_2121Sofosbuvir
Antiinfectives For Systemic Use
Hepatitis C virus | Acquired immunodeficiency syndrome
Zika virus
Paraiba
NA
Real-time PCR
Decrease (>1 Log10 (GE/ml))
Approved
27902933
DrugRepV_2122Sofosbuvir
Antiinfectives For Systemic Use
Hepatitis C virus | Acquired immunodeficiency syndrome
Zika virus
Paraiba
NA
Real-time PCR
Decrease (2 Log10 (GE/ml))
Approved
27902933
DrugRepV_2123Sofosbuvir
Antiinfectives For Systemic Use
Hepatitis C virus | Acquired immunodeficiency syndrome
Zika virus
Dakar
NA
Real-time PCR
Decrease (>1 Log10 (GE/ml))
Approved
27902933
DrugRepV_2124Sofosbuvir
Antiinfectives For Systemic Use
Hepatitis C virus | Acquired immunodeficiency syndrome
Zika virus
Dakar
NA
Real-time PCR
Decrease (>2 Log10 (GE/ml))
Approved
27902933
DrugRepV_2125Sofosbuvir
Antiinfectives For Systemic Use
Hepatitis C virus | Acquired immunodeficiency syndrome
Zika virus
Paraiba
NA
Flow cytometry
Decrease (50 %)
Approved
27902933
DrugRepV_2126Sofosbuvir
Antiinfectives For Systemic Use
Hepatitis C virus | Acquired immunodeficiency syndrome
Zika virus
Paraiba
NA
Flow cytometry
Decrease (50 %)
Approved
27902933
DrugRepV_2127Sofosbuvir
Antiinfectives For Systemic Use
Hepatitis C virus | Acquired immunodeficiency syndrome
Zika virus
Dakar/41519
NA
Survival assay
Increase
Approved
27902933
DrugRepV_2128Ribavirin
Antiinfectives For Systemic Use
Hepatitis C virus
Zika virus
MR766
NA
Cytopathic effect (CPE) assay
Decrease (50 %)
Approved
27163257
DrugRepV_2129Ribavirin
Antiinfectives For Systemic Use
Hepatitis C virus
Zika virus
MR766
NA
Virus yield reduction assay
Decrease (50 %)
Approved
27163257
DrugRepV_2198Neomycin Sulfate
Antiinfectives For Systemic Use
Bacterial infections
Chikungunya virus
vAc-CHIKV 26S-Rhir-E
NA
Fusion index-Fluorescent Intensities
No significant decrease (10.0220837 %)
Approved
27742486
DrugRepV_2200Rifampin
Antiinfectives For Systemic Use
Tuberculosis and Tuberculosis-related mycobacterial infections
Chikungunya virus
vAc-CHIKV 26S-Rhir-E
NA
Fusion index-Fluorescent Intensities
No significant decrease (9.11795232 %)
Approved
27742486
DrugRepV_2201Atazanavir Sulfate
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Chikungunya virus
vAc-CHIKV 26S-Rhir-E
NA
Fusion index-Fluorescent Intensities
No significant decrease (8.91119067 %)
Approved
27742486
DrugRepV_2210Pefloxacin Mesylate
Antiinfectives For Systemic Use
Gonococcal urethritis in males
Chikungunya virus
vAc-CHIKV 26S-Rhir-E
NA
Fusion index-Fluorescent Intensities
No significant decrease (7.83586814 %)
Approved
27742486
DrugRepV_2214Moroxydine
Antiinfectives For Systemic Use
Influenza
Chikungunya virus
vAc-CHIKV 26S-Rhir-E
NA
Fusion index-Fluorescent Intensities
No significant decrease (7.65475751 %)
Experimental
27742486
DrugRepV_2231Ribavirin
Antiinfectives For Systemic Use
Hepatitis C virus
Chikungunya virus
vAc-CHIKV 26S-Rhir-E
NA
Fusion index-Fluorescent Intensities
No significant decrease (6.95397975 %)
Approved
27742486
DrugRepV_2240Itraconazole
Antiinfectives For Systemic Use
Fungal infections (Pulmonary and extrapulmonary blastomycosis, Histoplasmosis, Aspergillosis, and Onychomycosis)
Chikungunya virus
vAc-CHIKV 26S-Rhir-E
NA
Fusion index-Fluorescent Intensities
No significant decrease (6.35827197 %)
Approved, Investigational
27742486
DrugRepV_2245Methenamine
Antiinfectives For Systemic Use
Urinary tract infection
Chikungunya virus
vAc-CHIKV 26S-Rhir-E
NA
Fusion index-Fluorescent Intensities
No significant decrease (6.11366498 %)
Approved, Vet approved
27742486
DrugRepV_2246Azithromycin
Antiinfectives For Systemic Use
Microbial infections
Chikungunya virus
vAc-CHIKV 26S-Rhir-E
NA
Fusion index-Fluorescent Intensities
No significant decrease (6.11366498 %)
Approved
27742486
DrugRepV_2258Biapenem
Antiinfectives For Systemic Use
Bacterial infections
Chikungunya virus
vAc-CHIKV 26S-Rhir-E
NA
Fusion index-Fluorescent Intensities
No significant decrease (5.72083061 %)
Investigational
27742486
DrugRepV_2263Idoxuridine
Antiinfectives For Systemic Use
Keratoconjunctivitis and Keratitis caused by herpes simplex virus
Chikungunya virus
vAc-CHIKV 26S-Rhir-E
NA
Fusion index-Fluorescent Intensities
No significant decrease (5.28034643 %)
Approved, Investigational
27742486
DrugRepV_2265Clindamycin Phosphate
Antiinfectives For Systemic Use
Bacterial infections
Chikungunya virus
vAc-CHIKV 26S-Rhir-E
NA
Fusion index-Fluorescent Intensities
No significant decrease (5.23907349 %)
Approved
27742486
DrugRepV_2269Tigecycline
Antiinfectives For Systemic Use
Complicated skin and skin structure infections
Chikungunya virus
vAc-CHIKV 26S-Rhir-E
NA
Fusion index-Fluorescent Intensities
No significant decrease (5.03969688 %)
Approved
27742486
DrugRepV_2282Doripenem Hydrate
Antiinfectives For Systemic Use
Intra-abdominal infections and complicated urinary tract infections
Chikungunya virus
vAc-CHIKV 26S-Rhir-E
NA
Fusion index-Fluorescent Intensities
No significant decrease (4.71564204 %)
Approved
27742486
DrugRepV_2283Sulfamethazine
Antiinfectives For Systemic Use
Bacterial infections (Bronchitis, prostatitis and urinary tract infections)
Chikungunya virus
vAc-CHIKV 26S-Rhir-E
NA
Fusion index-Fluorescent Intensities
No significant decrease (4.70881807 %)
Approved, Investigational, Vet approved
27742486
DrugRepV_2299Sulfapyridine
Antiinfectives For Systemic Use
Dermatitis herpetiformis | Benign mucous membrane pemphigoid | Pyoderma gangrenosum
Chikungunya virus
vAc-CHIKV 26S-Rhir-E
NA
Fusion index-Fluorescent Intensities
No significant decrease (4.40977237 %)
Approved
27742486
DrugRepV_2301Thiamphenicol
Antiinfectives For Systemic Use
Infectious diseases in cattle, pigs and poultry)
Chikungunya virus
vAc-CHIKV 26S-Rhir-E
NA
Fusion index-Fluorescent Intensities
No significant decrease (4.40312446 %)
Experimental, Investigational
27742486
DrugRepV_2310Sulfamethizole
Antiinfectives For Systemic Use
Urinary tract infection
Chikungunya virus
vAc-CHIKV 26S-Rhir-E
NA
Fusion index-Fluorescent Intensities
No significant decrease (4.08218845 %)
Approved, Investigational, Vet approved
27742486
DrugRepV_2313Ritonavir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Chikungunya virus
vAc-CHIKV 26S-Rhir-E
NA
Fusion index-Fluorescent Intensities
No significant decrease (3.98622242 %)
Approved, Investigational
27742486
DrugRepV_2314Lopinavir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Chikungunya virus
vAc-CHIKV 26S-Rhir-E
NA
Fusion index-Fluorescent Intensities
No significant decrease (3.96247894 %)
Approved
27742486
DrugRepV_2324Isoniazid
Antiinfectives For Systemic Use
Tuberculosis
Chikungunya virus
vAc-CHIKV 26S-Rhir-E
NA
Fusion index-Fluorescent Intensities
No significant decrease (3.74356574 %)
Approved, Investigational
27742486
DrugRepV_2328Ketoconazole
Antiinfectives For Systemic Use
Fungal infections
Chikungunya virus
vAc-CHIKV 26S-Rhir-E
NA
Fusion index-Fluorescent Intensities
No significant decrease (3.68563359 %)
Approved, Investigational
27742486
DrugRepV_2338Posaconazole
Antiinfectives For Systemic Use
Fungal infections (Aspergillus and Candida infections)
Chikungunya virus
vAc-CHIKV 26S-Rhir-E
NA
Fusion index-Fluorescent Intensities
No significant decrease (3.43393568 %)
Approved, Investigational, Vet approved
27742486
DrugRepV_2343Protionamide
Antiinfectives For Systemic Use
MDR-TB | Acquired immunodeficiency syndrome
Chikungunya virus
vAc-CHIKV 26S-Rhir-E
NA
Fusion index-Fluorescent Intensities
No significant decrease (3.29332873 %)
Approved, Investigational
27742486
DrugRepV_2347Amoxicillin Sodium
Antiinfectives For Systemic Use
Bacterial infections
Chikungunya virus
vAc-CHIKV 26S-Rhir-E
NA
Fusion index-Fluorescent Intensities
No significant decrease (3.26461637 %)
Approved
27742486
DrugRepV_2354Cephradine
Antiinfectives For Systemic Use
Bacterial infections
Chikungunya virus
vAc-CHIKV 26S-Rhir-E
NA
Fusion index-Fluorescent Intensities
No significant decrease (3.17042436 %)
Approved
27742486
DrugRepV_2358Sitafloxacin Hydrate
Antiinfectives For Systemic Use
Bacterial infections (respiratory and urinary tract infections)
Chikungunya virus
vAc-CHIKV 26S-Rhir-E
NA
Fusion index-Fluorescent Intensities
No significant decrease (2.96036077 %)
Experimental, Investigational
27742486
DrugRepV_2360Enoxacin
Antiinfectives For Systemic Use
Bacterial infections
Chikungunya virus
vAc-CHIKV 26S-Rhir-E
NA
Fusion index-Fluorescent Intensities
No significant decrease (2.93176568 %)
Approved
27742486
DrugRepV_2368Ampicillin Sodium
Antiinfectives For Systemic Use
Bacterial infections
Chikungunya virus
vAc-CHIKV 26S-Rhir-E
NA
Fusion index-Fluorescent Intensities
No significant decrease (2.75763916 %)
Approved
27742486
DrugRepV_2383Bacitracin Zinc
Antiinfectives For Systemic Use
Pneumonia and empyema
Chikungunya virus
vAc-CHIKV 26S-Rhir-E
NA
Fusion index-Fluorescent Intensities
No significant decrease (2.42855269 %)
Approved
27742486
DrugRepV_2403Clindamycin Hydrochloride
Antiinfectives For Systemic Use
Bacterial infections
Chikungunya virus
vAc-CHIKV 26S-Rhir-E
NA
Fusion index-Fluorescent Intensities
No significant decrease (2.19411786 %)
Approved
27742486
DrugRepV_2404Spectinomycin Hydrochloride
Antiinfectives For Systemic Use
Bacterial infections (Gonorrheal urethritis and proctitis)
Chikungunya virus
vAc-CHIKV 26S-Rhir-E
NA
Fusion index-Fluorescent Intensities
No significant decrease (2.18634054 %)
Approved, Investigational, Vet approved
27742486
DrugRepV_2424Sulfameter
Antiinfectives For Systemic Use
Leprosy | Urinary | Respiratory tract infections
Chikungunya virus
vAc-CHIKV 26S-Rhir-E
NA
Fusion index-Fluorescent Intensities
No significant decrease (1.81863222 %)
Approved
27742486
DrugRepV_2426Norfloxacin
Antiinfectives For Systemic Use
Urinary tract infection
Chikungunya virus
vAc-CHIKV 26S-Rhir-E
NA
Fusion index-Fluorescent Intensities
No significant decrease (1.69457675 %)
Approved
27742486
DrugRepV_2438Rimantadine
Antiinfectives For Systemic Use
Influenza A virus
Chikungunya virus
vAc-CHIKV 26S-Rhir-E
NA
Fusion index-Fluorescent Intensities
No significant decrease (1.43192971 %)
Approved, Investigational
27742486
DrugRepV_2439Rifapentine
Antiinfectives For Systemic Use
Tuberculosis
Chikungunya virus
vAc-CHIKV 26S-Rhir-E
NA
Fusion index-Fluorescent Intensities
No significant decrease (1.3653391 %)
Approved, Investigational
27742486
DrugRepV_2445Gatifloxacin
Antiinfectives For Systemic Use
Bacterial infections (Bronchitis, sinusitis, Community-acquired pneumonia, and Skin infections)
Chikungunya virus
vAc-CHIKV 26S-Rhir-E
NA
Fusion index-Fluorescent Intensities
No significant decrease (1.22310404 %)
Approved, Investigational
27742486
DrugRepV_2447Raltegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Chikungunya virus
vAc-CHIKV 26S-Rhir-E
NA
Fusion index-Fluorescent Intensities
No significant decrease (1.14736269 %)
Approved
27742486
DrugRepV_2448Cefoperazone
Antiinfectives For Systemic Use
Bacterial infections
Chikungunya virus
vAc-CHIKV 26S-Rhir-E
NA
Fusion index-Fluorescent Intensities
No significant decrease (1.13001149 %)
Approved
27742486
DrugRepV_2449Tetracycline Hydrochloride
Antiinfectives For Systemic Use
Bacterial infections (Rocky Mountain spotted fever | Typhus fever | Tick fevers | Q fever | Rickettsialpox | Brill-Zinsser disease)
Chikungunya virus
vAc-CHIKV 26S-Rhir-E
NA
Fusion index-Fluorescent Intensities
No significant decrease (1.08422039 %)
Approved, Vet approved
27742486
DrugRepV_2455Sulphadimethoxine
Antiinfectives For Systemic Use
Respiratory infection | Urinary tract infection | Enteric infection | Soft tissue infection
Chikungunya virus
vAc-CHIKV 26S-Rhir-E
NA
Fusion index-Fluorescent Intensities
No significant decrease (0.99278461 %)
Approved, Vet approved
27742486
DrugRepV_2457Amikacin Hydrate
Antiinfectives For Systemic Use
Bacterial infections
Chikungunya virus
vAc-CHIKV 26S-Rhir-E
NA
Fusion index-Fluorescent Intensities
No significant decrease (0.87227544 %)
Approved
27742486
DrugRepV_2459Pyrazinamide
Antiinfectives For Systemic Use
Tuberculosis
Chikungunya virus
vAc-CHIKV 26S-Rhir-E
NA
Fusion index-Fluorescent Intensities
No significant decrease (0.85917346 %)
Approved, Investigational
27742486
DrugRepV_2476Ethionamide
Antiinfectives For Systemic Use
Tuberculosis
Chikungunya virus
vAc-CHIKV 26S-Rhir-E
NA
Fusion index-Fluorescent Intensities
No significant decrease (0.45109184 %)
Approved
27742486
DrugRepV_2478Streptomycin Sulfate
Antiinfectives For Systemic Use
Tuberculosis | Tularemia | Plague | Brucellosis | Endocarditis
Chikungunya virus
vAc-CHIKV 26S-Rhir-E
NA
Fusion index-Fluorescent Intensities
No significant decrease (0.42772783 %)
Approved, Vet approved
27742486
DrugRepV_2486Cefditoren Pivoxil
Antiinfectives For Systemic Use
Bacterial infections
Chikungunya virus
vAc-CHIKV 26S-Rhir-E
NA
Fusion index-Fluorescent Intensities
No significant decrease (0.31336219 %)
Approved
27742486
DrugRepV_2510Maraviroc
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Chikungunya virus
vAc-CHIKV 26S-Rhir-E
NA
Fusion index-Fluorescent Intensities
Increase (-0.0137712 %)
Approved, Investigational
27742486
DrugRepV_2511Carbenicillin Disodium
Antiinfectives For Systemic Use
Urinary tract infection
Chikungunya virus
vAc-CHIKV 26S-Rhir-E
NA
Fusion index-Fluorescent Intensities
Increase (-0.0151285 %)
Approved
27742486
DrugRepV_2517Clarithromycin
Antiinfectives For Systemic Use
Microbial infections
Chikungunya virus
vAc-CHIKV 26S-Rhir-E
NA
Fusion index-Fluorescent Intensities
Increase (-0.1486584 %)
Approved
27742486
DrugRepV_2518Ganciclovir
Antiinfectives For Systemic Use
Cytomegalovirus infection
Chikungunya virus
vAc-CHIKV 26S-Rhir-E
NA
Fusion index-Fluorescent Intensities
Increase (-0.183847 %)
Approved, Investigational
27742486
DrugRepV_2530Moxifloxacin Hydrochloride
Antiinfectives For Systemic Use
Sinusitis | Pneumonia | Chronic bronchitis
Chikungunya virus
vAc-CHIKV 26S-Rhir-E
NA
Fusion index-Fluorescent Intensities
Increase (-0.5365847 %)
Approved, Investigational
27742486
DrugRepV_2531Meropenem
Antiinfectives For Systemic Use
Bacterial infections (Skin infection)
Chikungunya virus
vAc-CHIKV 26S-Rhir-E
NA
Fusion index-Fluorescent Intensities
Increase (-0.5411877 %)
Approved, Investigational
27742486
DrugRepV_2540Valacyclovir Hydrochloride
Antiinfectives For Systemic Use
Herpes simplex and Zoster virus
Chikungunya virus
vAc-CHIKV 26S-Rhir-E
NA
Fusion index-Fluorescent Intensities
Increase (-0.6677761 %)
Approved
27742486
DrugRepV_2543Cefaclor
Antiinfectives For Systemic Use
Bacterial infections
Chikungunya virus
vAc-CHIKV 26S-Rhir-E
NA
Fusion index-Fluorescent Intensities
Increase (-0.7251215 %)
Approved
27742486
DrugRepV_2546Ciprofloxacin
Antiinfectives For Systemic Use
Bacterial infections
Chikungunya virus
vAc-CHIKV 26S-Rhir-E
NA
Fusion index-Fluorescent Intensities
Increase (-0.8107955 %)
Approved
27742486
DrugRepV_2554Oxytetracycline dihydrate
Antiinfectives For Systemic Use
Bacterial infections
Chikungunya virus
vAc-CHIKV 26S-Rhir-E
NA
Fusion index-Fluorescent Intensities
Increase (-0.9136131 %)
Approved, Investigational, Vet approved
27742486
DrugRepV_2557Aztreonam
Antiinfectives For Systemic Use
Bacterial infections
Chikungunya virus
vAc-CHIKV 26S-Rhir-E
NA
Fusion index-Fluorescent Intensities
Increase (-0.9905633 %)
Approved
27742486
DrugRepV_2566Lincomycin Hydrochloride
Antiinfectives For Systemic Use
Bacterial infections
Chikungunya virus
vAc-CHIKV 26S-Rhir-E
NA
Fusion index-Fluorescent Intensities
Increase (-1.1874718 %)
Approved, Vet approved
27742486
DrugRepV_2568Oxacillin Sodium Monohydrate
Antiinfectives For Systemic Use
Staphylococci infections
Chikungunya virus
vAc-CHIKV 26S-Rhir-E
NA
Fusion index-Fluorescent Intensities
Increase (-1.2220202 %)
Approved, Investigational
27742486
DrugRepV_2569Entecavir Hydrate
Antiinfectives For Systemic Use
Hepatitis B virus
Chikungunya virus
vAc-CHIKV 26S-Rhir-E
NA
Fusion index-Fluorescent Intensities
Increase (-1.2373625 %)
Approved
27742486
DrugRepV_2575Amprenavir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Chikungunya virus
vAc-CHIKV 26S-Rhir-E
NA
Fusion index-Fluorescent Intensities
Increase (-1.2615469 %)
Approved
27742486
DrugRepV_2584Flumequine
Antiinfectives For Systemic Use
Bacterial infections
Chikungunya virus
vAc-CHIKV 26S-Rhir-E
NA
Fusion index-Fluorescent Intensities
Increase (-1.3882128 %)
Withdrawn
27742486
DrugRepV_2598Telbivudine
Antiinfectives For Systemic Use
Hepatitis B virus
Chikungunya virus
vAc-CHIKV 26S-Rhir-E
NA
Fusion index-Fluorescent Intensities
Increase (-1.5369604 %)
Approved
27742486
DrugRepV_2606Lomefloxacin Hydrochloride
Antiinfectives For Systemic Use
Bacterial infections (respiratory tract (chronic bronchitis) and urinary tract)
Chikungunya virus
vAc-CHIKV 26S-Rhir-E
NA
Fusion index-Fluorescent Intensities
Increase (-1.6544832 %)
Approved, Investigational
27742486
DrugRepV_2607Linezolid
Antiinfectives For Systemic Use
Bacterial infections
Chikungunya virus
vAc-CHIKV 26S-Rhir-E
NA
Fusion index-Fluorescent Intensities
Increase (-1.6567659 %)
Approved, Investigational
27742486
DrugRepV_2609Nevirapine
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Chikungunya virus
vAc-CHIKV 26S-Rhir-E
NA
Fusion index-Fluorescent Intensities
Increase (-1.6918978 %)
Approved
27742486
DrugRepV_2626Voriconazole
Antiinfectives For Systemic Use
Fungal infections
Chikungunya virus
vAc-CHIKV 26S-Rhir-E
NA
Fusion index-Fluorescent Intensities
Increase (-1.8244532 %)
Approved
27742486
DrugRepV_2640Levofloxacin
Antiinfectives For Systemic Use
Bacterial infections (Conjunctivitis)
Chikungunya virus
vAc-CHIKV 26S-Rhir-E
NA
Fusion index-Fluorescent Intensities
Increase (-2.028788 %)
Approved, Investigational
27742486
DrugRepV_2645Cidofovir
Antiinfectives For Systemic Use
Cytomegalovirus infection
Chikungunya virus
vAc-CHIKV 26S-Rhir-E
NA
Fusion index-Fluorescent Intensities
Increase (-2.1015434 %)
Approved
27742486
DrugRepV_2653Fluconazole
Antiinfectives For Systemic Use
Fungal infections
Chikungunya virus
vAc-CHIKV 26S-Rhir-E
NA
Fusion index-Fluorescent Intensities
Increase (-2.2384772 %)
Approved, Investigational
27742486
DrugRepV_2654Trimethoprim
Antiinfectives For Systemic Use
Urinary tract infections | Uncomplicated pyelonephritis (with sulfamethoxazole) | Mild acute prostatitis
Chikungunya virus
vAc-CHIKV 26S-Rhir-E
NA
Fusion index-Fluorescent Intensities
Increase (-2.2572502 %)
Approved
27742486
DrugRepV_2667Azlocillin Sodium salt
Antiinfectives For Systemic Use
Bacterial infections
Chikungunya virus
vAc-CHIKV 26S-Rhir-E
NA
Fusion index-Fluorescent Intensities
Increase (-2.4022354 %)
Approved
27742486
DrugRepV_2673Cefprozil Hydrate
Antiinfectives For Systemic Use
Bacterial infections
Chikungunya virus
vAc-CHIKV 26S-Rhir-E
NA
Fusion index-Fluorescent Intensities
Increase (-2.4845708 %)
Approved
27742486
DrugRepV_2685Oseltamivir phosphate
Antiinfectives For Systemic Use
Influenza A/B virus
Chikungunya virus
vAc-CHIKV 26S-Rhir-E
NA
Fusion index-Fluorescent Intensities
Increase (-2.6044621 %)
Approved
27742486
DrugRepV_2689Daptomycin
Antiinfectives For Systemic Use
Bacterial infections
Chikungunya virus
vAc-CHIKV 26S-Rhir-E
NA
Fusion index-Fluorescent Intensities
Increase (-2.764086 %)
Approved
27742486
DrugRepV_2693Cloxacillin Sodium
Antiinfectives For Systemic Use
Bacterial infections
Chikungunya virus
vAc-CHIKV 26S-Rhir-E
NA
Fusion index-Fluorescent Intensities
Increase (-2.8753795 %)
Approved
27742486
DrugRepV_2697Fleroxacin
Antiinfectives For Systemic Use
Bacterial infections
Chikungunya virus
vAc-CHIKV 26S-Rhir-E
NA
Fusion index-Fluorescent Intensities
Increase (-2.9243945 %)
Experimental
27742486
DrugRepV_2700Tenofovir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Chikungunya virus
vAc-CHIKV 26S-Rhir-E
NA
Fusion index-Fluorescent Intensities
Increase (-2.9691678 %)
Approved, Investigational
27742486
DrugRepV_2704Sulbactam Sodium
Antiinfectives For Systemic Use
Bacterial infections (Skin infection)
Chikungunya virus
vAc-CHIKV 26S-Rhir-E
NA
Fusion index-Fluorescent Intensities
Increase (-3.0092385 %)
Approved
27742486
DrugRepV_2706Sulfadiazine
Antiinfectives For Systemic Use
Rheumatic fever | Meningococcal meningitis
Chikungunya virus
vAc-CHIKV 26S-Rhir-E
NA
Fusion index-Fluorescent Intensities
Increase (-3.0259808 %)
Approved, Investigational, Vet approved
27742486
DrugRepV_2710D-Cycloserine
Antiinfectives For Systemic Use
Antibiotic
Chikungunya virus
vAc-CHIKV 26S-Rhir-E
NA
Fusion index-Fluorescent Intensities
Increase (-3.0661555 %)
Approved
27742486
DrugRepV_2720Tenofovir disoproxil Fumarate
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Chikungunya virus
vAc-CHIKV 26S-Rhir-E
NA
Fusion index-Fluorescent Intensities
Increase (-3.295385 %)
Approved, Investigational
27742486
DrugRepV_2721Adefovir dipivoxil
Antiinfectives For Systemic Use
Hepatitis B virus
Chikungunya virus
vAc-CHIKV 26S-Rhir-E
NA
Fusion index-Fluorescent Intensities
Increase (-3.3056399 %)
Approved
27742486
DrugRepV_2727Ofloxacin
Antiinfectives For Systemic Use
Respiratory tract infections | Kidney infection | Skin infection
Chikungunya virus
vAc-CHIKV 26S-Rhir-E
NA
Fusion index-Fluorescent Intensities
Increase (-3.4146475 %)
Approved
27742486
DrugRepV_2731Rifabutin
Antiinfectives For Systemic Use
Mycobacterium avium complex (MAC) disease in patients with advanced Acquired immunodeficiency syndrome infection
Chikungunya virus
vAc-CHIKV 26S-Rhir-E
NA
Fusion index-Fluorescent Intensities
Increase (-3.4674544 %)
Approved, Investigational
27742486
DrugRepV_2734Sulbactam
Antiinfectives For Systemic Use
Bacterial infections (Skin infection)
Chikungunya virus
vAc-CHIKV 26S-Rhir-E
NA
Fusion index-Fluorescent Intensities
Increase (-3.5031618 %)
Approved
27742486
DrugRepV_2737Didanosine
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Chikungunya virus
vAc-CHIKV 26S-Rhir-E
NA
Fusion index-Fluorescent Intensities
Increase (-3.5849038 %)
Approved
27742486
DrugRepV_2743Oxytetracycline
Antiinfectives For Systemic Use
Bacterial infections
Chikungunya virus
vAc-CHIKV 26S-Rhir-E
NA
Fusion index-Fluorescent Intensities
Increase (-3.6733944 %)
Approved, Investigational, Vet approved
27742486
DrugRepV_2764Zalcitabine
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome/AIDS
Chikungunya virus
vAc-CHIKV 26S-Rhir-E
NA
Fusion index-Fluorescent Intensities
Increase (-4.2270809 %)
Approved
27742486
DrugRepV_2775Flucytosine
Antiinfectives For Systemic Use
Fungal infections
Chikungunya virus
vAc-CHIKV 26S-Rhir-E
NA
Fusion index-Fluorescent Intensities
Increase (-4.4557163 %)
Approved, Investigational
27742486
DrugRepV_2777Sulfamerazine
Antiinfectives For Systemic Use
Bacterial infections (Bronchitis, prostatitis and urinary tract infections)
Chikungunya virus
vAc-CHIKV 26S-Rhir-E
NA
Fusion index-Fluorescent Intensities
Increase (-4.4815833 %)
Approved, Vet approved
27742486
DrugRepV_2783Elvitegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Chikungunya virus
vAc-CHIKV 26S-Rhir-E
NA
Fusion index-Fluorescent Intensities
Increase (-4.5754617 %)
Approved
27742486
DrugRepV_2791Abacavir Sulfate
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Chikungunya virus
vAc-CHIKV 26S-Rhir-E
NA
Fusion index-Fluorescent Intensities
Increase (-4.7456882 %)
Approved
27742486
DrugRepV_2795Roxithromycin
Antiinfectives For Systemic Use
Respiratory tract | Urinary and soft tissue infections
Chikungunya virus
vAc-CHIKV 26S-Rhir-E
NA
Fusion index-Fluorescent Intensities
Increase (-4.8220241 %)
Approved
27742486
DrugRepV_2801Lamivudine
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome | Hepatitis B virus
Chikungunya virus
vAc-CHIKV 26S-Rhir-E
NA
Fusion index-Fluorescent Intensities
Increase (-5.0142414 %)
Approved
27742486
DrugRepV_2833Etravirine
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Chikungunya virus
vAc-CHIKV 26S-Rhir-E
NA
Fusion index-Fluorescent Intensities
Increase (-5.947872 %)
Approved
27742486
DrugRepV_2839Emtricitabine
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Chikungunya virus
vAc-CHIKV 26S-Rhir-E
NA
Fusion index-Fluorescent Intensities
Increase (-6.2439742 %)
Approved
27742486
DrugRepV_2849Amikacin Sulfate
Antiinfectives For Systemic Use
Bacterial infections
Chikungunya virus
vAc-CHIKV 26S-Rhir-E
NA
Fusion index-Fluorescent Intensities
Increase (-6.6506378 %)
Approved
27742486
DrugRepV_2851Sulfamethoxazole
Antiinfectives For Systemic Use
Bacterial infections (Bronchitis, prostatitis and urinary tract infections)
Chikungunya virus
vAc-CHIKV 26S-Rhir-E
NA
Fusion index-Fluorescent Intensities
Increase (-6.7837639 %)
Approved
27742486
DrugRepV_2886Stavudine
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Chikungunya virus
vAc-CHIKV 26S-Rhir-E
NA
Fusion index-Fluorescent Intensities
Increase (-8.4649195 %)
Approved, Investigational
27742486
DrugRepV_2892Sparfloxacin
Antiinfectives For Systemic Use
Pneumonia | Acute bacterial exacerbations of chronic bronchitis
Chikungunya virus
vAc-CHIKV 26S-Rhir-E
NA
Fusion index-Fluorescent Intensities
Increase (-8.7240967 %)
Approved, Investigational, Withdrawn
27742486
DrugRepV_2901Amoxicillin
Antiinfectives For Systemic Use
Bacterial infections
Chikungunya virus
vAc-CHIKV 26S-Rhir-E
NA
Fusion index-Fluorescent Intensities
Increase (-9.1354562 %)
Approved
27742486
DrugRepV_2902Cefdinir
Antiinfectives For Systemic Use
Bacterial infections
Chikungunya virus
vAc-CHIKV 26S-Rhir-E
NA
Fusion index-Fluorescent Intensities
Increase (-9.1747501 %)
Approved
27742486
DrugRepV_2911Sulfanilamide
Antiinfectives For Systemic Use
Vulvovaginitis
Chikungunya virus
vAc-CHIKV 26S-Rhir-E
NA
Fusion index-Fluorescent Intensities
Increase (-9.7841731 %)
Approved
27742486
DrugRepV_2922Amphotericin B
Antiinfectives For Systemic Use
Fungal infections
Chikungunya virus
vAc-CHIKV 26S-Rhir-E
NA
Fusion index-Fluorescent Intensities
Increase (-11.133117 %)
Approved
27742486
DrugRepV_2933Erythromycin
Antiinfectives For Systemic Use
Bacterial infections
Chikungunya virus
vAc-CHIKV 26S-Rhir-E
NA
Fusion index-Fluorescent Intensities
Increase (-14.433754 %)
Approved
27742486
DrugRepV_2934Chloramphenicol
Antiinfectives For Systemic Use
Bacterial infections
Chikungunya virus
vAc-CHIKV 26S-Rhir-E
NA
Fusion index-Fluorescent Intensities
Increase (-14.926902 %)
Approved
27742486
DrugRepV_2952Tetracycline
Antiinfectives For Systemic Use
Bacterial infections (Rocky Mountain spotted fever | Typhus fever | Tick fevers | Q fever | Rickettsialpox | Brill-Zinsser disease)
Chikungunya virus
Clinical isolate of CHIKV (East/Central/South African genotype)
NA
Plaque assay
Decrease (2.76 ÌÑ 107 pfu/ml)
Approved
25970853
DrugRepV_2953Doxycycline
Antiinfectives For Systemic Use
Bacterial infections
Chikungunya virus
Clinical isolate of CHIKV (East/Central/South African genotype)
NA
Plaque assay
Decrease (1.50 ÌÑ 107 pfu/ml)
Approved
25970853
DrugRepV_2954Rolitetracycline
Antiinfectives For Systemic Use
Bacterial infection
Chikungunya virus
Clinical isolate of CHIKV (East/Central/South African genotype)
NA
Plaque assay
Decrease (3.76 ÌÑ 107 pfu/ml)
Approved
25970853
DrugRepV_2955Ribavirin
Antiinfectives For Systemic Use
Hepatitis C virus
Chikungunya virus
Clinical isolate of CHIKV (East/Central/South African genotype)
NA
Plaque assay
Decrease (0.96 ÌÑ 107 pfu/ml)
Approved
25970853
DrugRepV_2956Aciclovir
Antiinfectives For Systemic Use
Viral infection
Chikungunya virus
Clinical isolate of CHIKV (East/Central/South African genotype)
NA
Plaque assay
Decrease (2.30 ÌÑ 107 pfu/ml)
Approved
25970853
DrugRepV_2957Doxycycline
Antiinfectives For Systemic Use
Bacterial infections
Chikungunya virus
Clinical isolate of CHIKV (East/Central/South African genotype)
NA
NA
NA
Approved
25970853
DrugRepV_2958Doxycycline
Antiinfectives For Systemic Use
Bacterial infections
Chikungunya virus
Clinical isolate of CHIKV (East/Central/South African genotype)
NA
NA
NA
Approved
25970853
DrugRepV_2959Doxycycline
Antiinfectives For Systemic Use
Bacterial infections
Chikungunya virus
Clinical isolate of CHIKV (East/Central/South African genotype)
NA
Enzyme-linked immunosorbent assay
Decrease (50 %)
Approved
25970853
DrugRepV_2960Ribavirin
Antiinfectives For Systemic Use
Hepatitis C virus
Chikungunya virus
Clinical isolate of CHIKV (East/Central/South African genotype)
NA
Enzyme-linked immunosorbent assay
Decrease (50 %)
Approved
25970853
DrugRepV_2962Doxycycline
Antiinfectives For Systemic Use
Bacterial infections
Chikungunya virus
Clinical isolate of CHIKV (East/Central/South African genotype)
NA
Enzyme-linked immunosorbent assay
Decrease (51 %)
Approved
25970853
DrugRepV_2963Ribavirin
Antiinfectives For Systemic Use
Hepatitis C virus
Chikungunya virus
Clinical isolate of CHIKV (East/Central/South African genotype)
NA
Enzyme-linked immunosorbent assay
Decrease (68 %)
Approved
25970853
DrugRepV_2965Doxycycline
Antiinfectives For Systemic Use
Bacterial infections
Chikungunya virus
Clinical isolate of CHIKV (East/Central/South African genotype)
NA
Plaque assay
Decrease (68 %)
Approved
25970853
DrugRepV_2966Ribavirin
Antiinfectives For Systemic Use
Hepatitis C virus
Chikungunya virus
Clinical isolate of CHIKV (East/Central/South African genotype)
NA
Plaque assay
Decrease (45 %)
Approved
25970853
DrugRepV_2968Doxycycline
Antiinfectives For Systemic Use
Bacterial infections
Chikungunya virus
Clinical isolate of CHIKV (East/Central/South African genotype)
NA
Plaque assay
Decrease (71 %)
Approved
25970853
DrugRepV_2969Ribavirin
Antiinfectives For Systemic Use
Hepatitis C virus
Chikungunya virus
Clinical isolate of CHIKV (East/Central/South African genotype)
NA
Plaque assay
Decrease (44 %)
Approved
25970853
DrugRepV_2971Doxycycline
Antiinfectives For Systemic Use
Bacterial infections
Chikungunya virus
Clinical isolate of CHIKV (East/Central/South African genotype)
NA
Plaque assay
Decrease (43 %)
Approved
25970853
DrugRepV_2972Ribavirin
Antiinfectives For Systemic Use
Hepatitis C virus
Chikungunya virus
Clinical isolate of CHIKV (East/Central/South African genotype)
NA
Plaque assay
Decrease (67 %)
Approved
25970853
DrugRepV_2974Doxycycline
Antiinfectives For Systemic Use
Bacterial infections
Chikungunya virus
Clinical isolate of CHIKV (East/Central/South African genotype)
NA
MTT assay
Decrease (65 %)
Approved
25970853
DrugRepV_2975Ribavirin
Antiinfectives For Systemic Use
Hepatitis C virus
Chikungunya virus
Clinical isolate of CHIKV (East/Central/South African genotype)
NA
MTT assay
Decrease (71.6 %)
Approved
25970853
DrugRepV_2982Ribavirin
Antiinfectives For Systemic Use
Hepatitis C virus
Chikungunya virus
CHIKV replicon
NA
EGFP assay
Decrease (50 %)
Approved
22205980
DrugRepV_2991Ribavirin
Antiinfectives For Systemic Use
Hepatitis C virus
Chikungunya virus
CHIKV replicon
NA
Rluc assay
Decrease (50 %)
Approved
22205980
DrugRepV_3051Amphotericin B
Antiinfectives For Systemic Use
Fungal infection
Chikungunya virus
CHIKV-Rluc
NA
Luciferase reporter assay
Decrease (77 %)
Approved
26752081
DrugRepV_3060Efavirenz
Antiinfectives For Systemic Use
Acquired immuno deficiency syndrome
Chikungunya virus
CHIKV-Rluc
NA
Luciferase reporter assay
Decrease (10 %)
Approved
26752081
DrugRepV_3062Amphotericin B
Antiinfectives For Systemic Use
Fungal infection
Chikungunya virus
CHIKV-Rluc
NA
Renilla luciferase assay
No significant effect (90 %)
Approved
26752081
DrugRepV_3156Ribavirin
Antiinfectives For Systemic Use
Hepatitis C virus
Chikungunya virus
Ross C347
NA
Cytopathic effect (CPE) assay
Decrease (50 %)
Approved
14670584
DrugRepV_3164Ribavirin
Antiinfectives For Systemic Use
Hepatitis C virus
Chikungunya virus
Ross C347
NA
Cytopathic effect (CPE) assay
Decrease (1.8 Log)
Approved
14670584
DrugRepV_3168Ribavirin
Antiinfectives For Systemic Use
Hepatitis C virus
Chikungunya virus
Ross C347
NA
Cytopathic effect (CPE) assay
Decrease (99 %)
Approved
14670584
DrugRepV_3190Rimantadine
Antiinfectives For Systemic Use
Influenza A virus
Influenza virus
A/Aichi/2/68
Pathway
Plaque assay
Decrease (50 %)
Approved, Investigational
22028179
DrugRepV_3193Rimantadine
Antiinfectives For Systemic Use
Influenza A virus
Influenza virus
A/Aichi/2/68
Pathway
Plaque assay
No significant reduction (No significant reduction log)
Approved, Investigational
22028179
DrugRepV_3196Rimantadine
Antiinfectives For Systemic Use
Influenza A virus
Influenza virus
A/Aichi/2/68
Pathway
Quantal assay
Decrease (1 log)
Approved, Investigational
22028179
DrugRepV_3349Oseltamivir
Antiinfectives For Systemic Use
Influenza A/B virus
Influenza virus
WSN/H1N1
Pathway
Plaque assay
No significant effect (40 %)
Approved
29990517
DrugRepV_3351Oseltamivir
Antiinfectives For Systemic Use
Influenza A/B virus
Influenza virus
WSN/H1N1
Pathway
Plaque assay
Decrease (1.5 Log)
Approved
29990517
DrugRepV_3370Ribavirin
Antiinfectives For Systemic Use
Hepatitis C virus
Influenza virus
A/ WSN/1933 (H1N1)
Pathway
High-throughput screening
Decrease (50 %)
Approved
24096239
DrugRepV_3377Ribavirin
Antiinfectives For Systemic Use
Hepatitis C virus
Middle East respiratory syndrome coronavirus
NA
NA
CPE inhibition assay
Decrease (50 %)
Approved
24096239
DrugRepV_3384Ribavirin
Antiinfectives For Systemic Use
Hepatitis C virus
Middle East respiratory syndrome coronavirus
NA
NA
CPE inhibition assay
Decrease (90 %)
Approved
24096239
DrugRepV_3390Ribavirin
Antiinfectives For Systemic Use
Hepatitis C virus
Middle East respiratory syndrome coronavirus
NA
NA
CPE inhibition assay
Decrease (99 %)
Approved
24096239
DrugRepV_3396Ribavirin
Antiinfectives For Systemic Use
Hepatitis C virus
Middle East respiratory syndrome coronavirus
NA
NA
Real-time PCR
Decrease (>2 Log)
Approved
24096239
DrugRepV_3402Ribavirin
Antiinfectives For Systemic Use
Hepatitis C virus
Middle East respiratory syndrome coronavirus
NA
NA
Plaque assay
Decrease (100 %)
Approved
24096239
DrugRepV_3410Etravirine
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Influenza virus
A/California/07/2009 (H1N1)
Pathway
Plaque assay
Decrease (50 %)
Approved
28778830
DrugRepV_3411Rilpivirine
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Influenza virus
A/California/07/2009 (H1N1)
Pathway
Plaque assay
Decrease (50 %)
Approved
28778830
DrugRepV_3412Oseltamivir
Antiinfectives For Systemic Use
Influenza A/B virus
Influenza virus
A/California/07/2009 (H1N1)
Pathway
Plaque assay
Decrease (50 %)
Approved
28778830
DrugRepV_3414Etravirine
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Influenza virus
B/Bris/60/2008 (Victoria)
Pathway
Plaque assay
Decrease (50 %)
Approved
28778830
DrugRepV_3415Oseltamivir
Antiinfectives For Systemic Use
Influenza A/B virus
Influenza virus
B/Bris/60/2008 (Victoria)
Pathway
Plaque assay
Decrease (50 %)
Approved
28778830
DrugRepV_3418Oseltamivir
Antiinfectives For Systemic Use
Influenza A/B virus
Influenza virus
A/California/7/2009 (H1N1)
Pathway
Plaque assay
Decrease (1.7 Log)
Approved
28778830
DrugRepV_3419Oseltamivir
Antiinfectives For Systemic Use
Influenza A/B virus
Influenza virus
A/California/7/2009 (H1N1)
Pathway
Plaque assay
Decrease (2 Log)
Approved
28778830
DrugRepV_3421Oseltamivir
Antiinfectives For Systemic Use
Influenza A/B virus
Influenza virus
A/WSN/1933 (H1N1)
Pathway
Plaque assay
Decrease (1.4 Log)
Approved
28778830
DrugRepV_3550Sofosbuvir
Antiinfectives For Systemic Use
Hepatitis C virus | Acquired immunodeficiency syndrome
Chikungunya virus
Asian strain
NA
Real-time PCR
Decrease (50 %)
Approved
30455237
DrugRepV_3551Sofosbuvir
Antiinfectives For Systemic Use
Hepatitis C virus | Acquired immunodeficiency syndrome
Chikungunya virus
Asian strain
NA
Yield reduction assay
Decrease (50 %)
Approved
30455237
DrugRepV_3552Ribavirin
Antiinfectives For Systemic Use
Hepatitis C virus
Chikungunya virus
Asian strain
NA
Real-time PCR
Decrease (50 %)
Approved
30455237
DrugRepV_3553Ribavirin
Antiinfectives For Systemic Use
Hepatitis C virus
Chikungunya virus
Asian strain
NA
Yield reduction assay
Decrease (50 %)
Approved
30455237
DrugRepV_3556Sofosbuvir
Antiinfectives For Systemic Use
Hepatitis C virus | Acquired immunodeficiency syndrome
Chikungunya virus
Asian strain
NA
Survival assay
Increase
Approved
30455237
DrugRepV_3557Ribavirin
Antiinfectives For Systemic Use
Hepatitis C virus
Chikungunya virus
181/clone 25
NA
Plaque assay
Decrease (50 %)
Approved
30354193
DrugRepV_3558Ribavirin
Antiinfectives For Systemic Use
Hepatitis C virus
Chikungunya virus
181/clone 25
NA
Plaque assay
Decrease (50 %)
Approved
30354193
DrugRepV_3559Ribavirin
Antiinfectives For Systemic Use
Hepatitis C virus
Chikungunya virus
181/clone 25
NA
Plaque assay
Decrease (50 %)
Approved
30354193
DrugRepV_3614Ribavirin
Antiinfectives For Systemic Use
Hepatitis C virus
Nipah virus
NA
NA
RT-PCR
Decrease
Approved
16641448
DrugRepV_3620Ribavirin
Antiinfectives For Systemic Use
Hepatitis C virus
Nipah virus
NA
NA
RT-PCR
Decrease
Approved
16641448
DrugRepV_3622Ribavirin
Antiinfectives For Systemic Use
Hepatitis C virus
Nipah virus
NA
NA
RT-PCR
Decrease
Approved
16641448
DrugRepV_3697Ribavirin
Antiinfectives For Systemic Use
Hepatitis C virus
Marburg virus
NA
NA
Luciferase assay
Decrease (50 %)
Approved
24713118
DrugRepV_3700Ribavirin
Antiinfectives For Systemic Use
Hepatitis C virus
Ebola virus
NA
NA
Luciferase assay
Decrease (50 %)
Approved
24713118
DrugRepV_3703Ribavirin
Antiinfectives For Systemic Use
Hepatitis C virus
Marburg virus
NA
NA
NA
Decrease (83 %)
Approved
24713118
DrugRepV_3707Ribavirin
Antiinfectives For Systemic Use
Hepatitis C virus
Ebola virus
NA
NA
NA
Decrease (0 %)
Approved
24713118
DrugRepV_3875Ribavirin
Antiinfectives For Systemic Use
Hepatitis C virus
Zika virus
Puerto Rican PRVABC-59
NA
Cytopathic effect (CPE) assay
Decrease (50 %)
Approved
27838352
DrugRepV_3876Ribavirin
Antiinfectives For Systemic Use
Hepatitis C virus
Zika virus
Puerto Rican PRVABC-59
NA
Cytopathic effect (CPE) assay
Decrease (50 %)
Approved
27838352
DrugRepV_3877Ribavirin
Antiinfectives For Systemic Use
Hepatitis C virus
Zika virus
Puerto Rican PRVABC-59
NA
Cytopathic effect (CPE) assay
Decrease (50 %)
Approved
27838352
DrugRepV_3878Ribavirin
Antiinfectives For Systemic Use
Hepatitis C virus
Zika virus
Malaysian P 6-740
NA
Cytopathic effect (CPE) assay
Decrease (50 %)
Approved
27838352
DrugRepV_3879Ribavirin
Antiinfectives For Systemic Use
Hepatitis C virus
Zika virus
Malaysian P 6-740
NA
Cytopathic effect (CPE) assay
Decrease (50 %)
Approved
27838352
DrugRepV_3880Ribavirin
Antiinfectives For Systemic Use
Hepatitis C virus
Zika virus
Ugandan MR-766
NA
Cytopathic effect (CPE) assay
Decrease (50 %)
Approved
27838352
DrugRepV_3881Ribavirin
Antiinfectives For Systemic Use
Hepatitis C virus
Zika virus
Ugandan MR-766
NA
Cytopathic effect (CPE) assay
Decrease (50 %)
Approved
27838352
DrugRepV_3882Ribavirin
Antiinfectives For Systemic Use
Hepatitis C virus
Zika virus
Ugandan MR-766
NA
Cytopathic effect (CPE) assay
Decrease (50 %)
Approved
27838352
DrugRepV_4301Ribavirin
Antiinfectives For Systemic Use
Hepatitis C virus
Chikungunya virus
NA
NA
NA
Decrease (50 %)
Approved
27460167
DrugRepV_4310Ribavirin
Antiinfectives For Systemic Use
Hepatitis C virus
Ebola virus
Mayinga
NA
MTT assay
Decrease (50 %)
Approved
9988190
DrugRepV_4313Ribavirin
Antiinfectives For Systemic Use
Hepatitis C virus
Ebola virus
Sudan (Boneface strain)
NA
Plaque reduction assay
Decrease (50 %)
Approved
9988190
DrugRepV_4515Ribavirin
Antiinfectives For Systemic Use
Hepatitis C virus
Influenza virus
NA
Pathway
NA
Decrease (50 %)
Approved
15200845
DrugRepV_4516Zanamivir
Antiinfectives For Systemic Use
Influenza virus
Influenza virus
NA
Pathway
NA
Decrease (50 %)
Approved
15200845
DrugRepV_4517Oseltamivir
Antiinfectives For Systemic Use
Influenza A/B virus
Influenza virus
NA
Pathway
NA
Decrease (50 %)
Approved
15200845
DrugRepV_4529Ganciclovir
Antiinfectives For Systemic Use
Cytomegalovirus infection
Severe acute respiratory syndrome coronavirus
NA
NA
CPE inhibition assay
Decrease
Approved, Investigational
15200845
DrugRepV_4530Ribavirin
Antiinfectives For Systemic Use
Hepatitis C virus
Severe acute respiratory syndrome coronavirus
NA
NA
CPE inhibition assay
Decrease (100 %)
Approved
15200845
DrugRepV_4531Indinavir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Severe acute respiratory syndrome coronavirus
NA
NA
CPE inhibition assay
Decrease
Approved
15200845
DrugRepV_4532Nelfinavir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Severe acute respiratory syndrome coronavirus
NA
NA
CPE inhibition assay
Decrease
Approved
15200845
DrugRepV_4533Saquinavir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Severe acute respiratory syndrome coronavirus
NA
NA
CPE inhibition assay
Decrease
Approved, Investigational
15200845
DrugRepV_4534Lamivudine
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome | Hepatitis B virus
Severe acute respiratory syndrome coronavirus
NA
NA
CPE inhibition assay
Decrease
Approved
15200845
DrugRepV_4535Zidovudine
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome/AIDS
Severe acute respiratory syndrome coronavirus
NA
NA
CPE inhibition assay
Decrease
Approved
15200845
DrugRepV_4536Oseltamivir
Antiinfectives For Systemic Use
Influenza A/B virus
Severe acute respiratory syndrome coronavirus
NA
NA
CPE inhibition assay
Decrease
Approved
15200845
DrugRepV_4537Zanamivir
Antiinfectives For Systemic Use
Influenza virus
Severe acute respiratory syndrome coronavirus
NA
NA
CPE inhibition assay
Decrease
Approved
15200845
DrugRepV_4539Foscarnet
Antiinfectives For Systemic Use
Cytomegalovirus retinitis | Herpesviruses | Acquired immunodeficiency syndrome
Severe acute respiratory syndrome coronavirus
NA
NA
CPE inhibition assay
Decrease
Approved
15200845
DrugRepV_4544Ribavirin
Antiinfectives For Systemic Use
Hepatitis C virus
Severe acute respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
Approved
15961169
DrugRepV_4545AZT
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Severe acute respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
Approved
15961169
DrugRepV_4546Lopinavir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Severe acute respiratory syndrome coronavirus
NA
NA
NA
Decrease (50 %)
Approved
15961169
DrugRepV_4614Ribavirin
Antiinfectives For Systemic Use
Hepatitis C virus
Severe acute respiratory syndrome coronavirus
v2163
NA
Cytopathic effect (CPE) assay
Decrease (50 %)
Approved
19853271
DrugRepV_4615Ribavirin
Antiinfectives For Systemic Use
Hepatitis C virus
Severe acute respiratory syndrome coronavirus
Urbani
NA
Cytopathic effect (CPE) assay
Decrease (50 %)
Approved
19853271
DrugRepV_4630Ribavirin
Antiinfectives For Systemic Use
Hepatitis C virus
Severe acute respiratory syndrome coronavirus
v2163
NA
Survival assay
No significant effect
Approved
19853271
DrugRepV_4648Sofosbuvir
Antiinfectives For Systemic Use
Hepatitis C virus | Acquired immunodeficiency syndrome
Zika virus
NA
NA
Plaque assay
Decrease (50 %)
Approved
28098253
DrugRepV_4649Ribavirin
Antiinfectives For Systemic Use
Hepatitis C virus
Zika virus
NA
NA
Plaque assay
Decrease (50 %)
Approved
28098253
DrugRepV_4651Sofosbuvir
Antiinfectives For Systemic Use
Hepatitis C virus | Acquired immunodeficiency syndrome
Zika virus
NA
NA
Plaque assay
Decrease (1.00E+02 pfu/ml)
Approved
28098253
DrugRepV_4652Sofosbuvir
Antiinfectives For Systemic Use
Hepatitis C virus | Acquired immunodeficiency syndrome
Zika virus
NA
NA
Plaque assay
Decrease (5.00E+07 pfu/ml)
Approved
28098253
DrugRepV_4688Ribavirin
Antiinfectives For Systemic Use
Hepatitis C virus
Zika virus
NA
NA
Phenotypic assay
Decrease (50 %)
Approved
30061280
DrugRepV_4692Sofosbuvir
Antiinfectives For Systemic Use
Hepatitis C virus | Acquired immunodeficiency syndrome
Zika virus
NA
NA
Phenotypic assay
Decrease (50 %)
Approved
30061280
DrugRepV_4709Ribavirin
Antiinfectives For Systemic Use
Hepatitis C virus
Zika virus
NA
NA
Immunoflourescence assay
Decrease
Approved
30061280
DrugRepV_4778Ribavirin
Antiinfectives For Systemic Use
Hepatitis C virus
Middle East respiratory syndrome coronavirus
Hu/Jordan-N3/2012
NA
Virus yield reduction assay
Decrease (30 %)
Approved
24323636
DrugRepV_4822Teicoplanin
Antiinfectives For Systemic Use
Bacterial infections
Ebola virus
NA
NA
Luciferase assay
Decrease (50 %)
Approved
26953343
DrugRepV_4823Teicoplanin
Antiinfectives For Systemic Use
Bacterial infections
Ebola virus
NA
NA
Luciferase assay
Decrease (50 %)
Approved
26953343
DrugRepV_4824Dalbavancin
Antiinfectives For Systemic Use
Bacterial infections
Ebola virus
NA
NA
Luciferase assay
Decrease (50 %)
Approved
26953343
DrugRepV_4825Oritavancin
Antiinfectives For Systemic Use
Acute bacterial skin | Skin structure infections
Ebola virus
NA
NA
Luciferase assay
Decrease (50 %)
Approved
26953343
DrugRepV_4826Telavancin
Antiinfectives For Systemic Use
Skin infections (Bacterial)
Ebola virus
NA
NA
Luciferase assay
Decrease (50 %)
Approved
26953343
DrugRepV_4829Teicoplanin
Antiinfectives For Systemic Use
Bacterial infections
Middle East respiratory syndrome coronavirus
NA
NA
Luciferase assay
Decrease (50 %)
Approved
26953343
DrugRepV_4830Dalbavancin
Antiinfectives For Systemic Use
Bacterial infections
Middle East respiratory syndrome coronavirus
NA
NA
Luciferase assay
Decrease (50 %)
Approved
26953343
DrugRepV_4831Oritavancin
Antiinfectives For Systemic Use
Acute bacterial skin | Skin structure infections
Middle East respiratory syndrome coronavirus
NA
NA
Luciferase assay
Decrease (50 %)
Approved
26953343
DrugRepV_4832Telavancin
Antiinfectives For Systemic Use
Skin infections (Bacterial)
Middle East respiratory syndrome coronavirus
NA
NA
Luciferase assay
Decrease (50 %)
Approved
26953343
DrugRepV_5078Ribavirin
Antiinfectives For Systemic Use
Hepatitis C virus
Crimean-Congo hemorrhagic fever virus
10200
NA
Survival assay
No significant effect
Approved
29936152
DrugRepV_5079Ribavirin
Antiinfectives For Systemic Use
Hepatitis C virus
Crimean-Congo hemorrhagic fever virus
Hoti
NA
Survival assay
No significant effect
Approved
29936152
DrugRepV_5080Ribavirin
Antiinfectives For Systemic Use
Hepatitis C virus
Crimean-Congo hemorrhagic fever virus
10200
NA
Real-time PCR
Decrease
Approved
29936152
DrugRepV_5081Ribavirin
Antiinfectives For Systemic Use
Hepatitis C virus
Crimean-Congo hemorrhagic fever virus
Hoti
NA
Real-time PCR
Decrease
Approved
29936152
DrugRepV_5082Ribavirin
Antiinfectives For Systemic Use
Hepatitis C virus
Crimean-Congo hemorrhagic fever virus
NA
NA
Real-time PCR
Decrease (100 Copies/ml)
Approved
29584885
DrugRepV_5098Ribavirin
Antiinfectives For Systemic Use
Hepatitis C virus
Crimean-Congo hemorrhagic fever virus
CCHFV/ZsG
NA
Fluorescence-based assay
Decrease (50 %)
Approved
29024765
DrugRepV_5120ABT-333
Antiinfectives For Systemic Use
Hepatitis C virus
Crimean-Congo hemorrhagic fever virus
CCHFV/ZsG
NA
Fluorescence-based assay
No significant effect (39 %)
Approved
29024765
DrugRepV_5125Lamivudine
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome | Hepatitis B virus
Crimean-Congo hemorrhagic fever virus
CCHFV/ZsG
NA
Fluorescence-based assay
No significant effect (24 %)
Approved
29024765
DrugRepV_5132PSI-7977
Antiinfectives For Systemic Use
Hepatitis C virus
Crimean-Congo hemorrhagic fever virus
CCHFV/ZsG
NA
Fluorescence-based assay
No significant effect (4 %)
Approved
29024765
DrugRepV_5136Ribavirin
Antiinfectives For Systemic Use
Hepatitis C virus
Crimean-Congo hemorrhagic fever virus
CCHFV/ZsG
NA
Fluorescence-based assay
No significant effect (2 %)
Approved
29024765
DrugRepV_5137Stavudine
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Crimean-Congo hemorrhagic fever virus
CCHFV/ZsG
NA
Fluorescence-based assay
No significant effect (26 %)
Approved, Investigational
29024765
DrugRepV_5139Tenofovir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Crimean-Congo hemorrhagic fever virus
CCHFV/ZsG
NA
Fluorescence-based assay
No significant effect (0 %)
Approved, Investigational
29024765
DrugRepV_5140Zidovudine
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome/AIDS
Crimean-Congo hemorrhagic fever virus
CCHFV/ZsG
NA
Fluorescence-based assay
No significant effect (27 %)
Approved
29024765
DrugRepV_5184Ribavirin
Antiinfectives For Systemic Use
Hepatitis C virus
Rift Valley fever virus
ZH501
NA
Immunoflourescence assay
Decrease (50 %)
Approved
25144302
DrugRepV_5190Ribavirin
Antiinfectives For Systemic Use
Hepatitis C virus
Rift Valley fever virus
ZH501
NA
Immunoflourescence assay
Decrease (50 %)
Approved
25144302
DrugRepV_5196Ribavirin
Antiinfectives For Systemic Use
Hepatitis C virus
Ebola virus
Zaire
NA
Immunoflourescence assay
Decrease (50 %)
Approved
25144302
DrugRepV_5201Ribavirin
Antiinfectives For Systemic Use
Hepatitis C virus
Marburg virus
Ci67
NA
Immunoflourescence assay
Decrease (50 %)
Approved
25144302
DrugRepV_5205Ribavirin
Antiinfectives For Systemic Use
Hepatitis C virus
Lassa virus
Josiah
NA
Immunoflourescence assay
Decrease (50 %)
Approved
25144302
DrugRepV_5219Ribavirin
Antiinfectives For Systemic Use
Hepatitis C virus
Rift Valley fever virus
RVF-VLPs
NA
RLuc expression
Decrease (87.2 %)
Approved
21994655
DrugRepV_5225Ribavirin
Antiinfectives For Systemic Use
Hepatitis C virus
Crimean-Congo hemorrhagic fever virus
IbAr 10200
NA
Neutral red uptake assay
Decrease (50 %)
Approved
15026198
DrugRepV_5230Ribavirin
Antiinfectives For Systemic Use
Hepatitis C virus
Crimean-Congo hemorrhagic fever virus
Spu 128/81
NA
Neutral red uptake assay
Decrease (50 %)
Approved
15026198
DrugRepV_5235Ribavirin
Antiinfectives For Systemic Use
Hepatitis C virus
Crimean-Congo hemorrhagic fever virus
Hy-13
NA
Neutral red uptake assay
Decrease (50 %)
Approved
15026198
DrugRepV_5240Ribavirin
Antiinfectives For Systemic Use
Hepatitis C virus
Crimean-Congo hemorrhagic fever virus
UG3010
NA
Neutral red uptake assay
Decrease (50 %)
Approved
15026198
DrugRepV_5252Rifampicin
Antiinfectives For Systemic Use
Tuberculosis and Tuberculosis-related mycobacterial infections
Variola virus
Butler
NA
Plaque assay
Decrease (Complete inhibition Plaque size)
Approved
4321450
DrugRepV_5475Penciclovir
Antiinfectives For Systemic Use
Recurrent cold sores on the lips and face from Herpesvirus invections
SARS Coronavirus-2
nCoV- 2019BetaCoV/Wuhan/WIV04/2019
NA
qRT-PCR
Decrease (50 %)
Approved
32020029
DrugRepV_5524Ribavirin
Antiinfectives For Systemic Use
Hepatitis C virus
Lassa virus
NA
NA
Gaussia luciferase (Gluc) Glow assay
Decrease (50 %)
Approved
31786250
DrugRepV_5551Ribavirin
Antiinfectives For Systemic Use
Hepatitis C virus
SARS Coronavirus-2
2019-nCoV/USA-WA1/2020
NA
NA
Decrease (50 %)
Approved
32353859
DrugRepV_5591Chloramphenicol
Antiinfectives For Systemic Use
Bacterial infections
SARS Coronavirus-2
2019-nCoV/USA-WA1/2020
NA
NA
Decrease (50 %)
Approved
32353859
DrugRepV_5592Tigecycline
Antiinfectives For Systemic Use
Complicated skin and skin structure infections
SARS Coronavirus-2
2019-nCoV/USA-WA1/2020
NA
NA
Decrease (50 %)
Approved
32353859
DrugRepV_5593Linezolid
Antiinfectives For Systemic Use
Bacterial infections
SARS Coronavirus-2
2019-nCoV/USA-WA1/2020
NA
NA
Decrease (50 %)
Approved, Investigational
32353859
DrugRepV_5628Minocycline
Antiinfectives For Systemic Use
Rocky Mountain spotted fever | Typhus fever and the typhus group | Q fever | Rickettsial pox | tick fevers caused by Rickettsiae | Upper respiratory tract infections caused by Streptococcus pneumoniae
Dengue virus
16681
Pathway
Enzyme-linked immunosorbent assay
Decrease (20 %)
Approved, Investigational
27396621
DrugRepV_5629Minocycline
Antiinfectives For Systemic Use
Rocky Mountain spotted fever | Typhus fever and the typhus group | Q fever | Rickettsial pox | tick fevers caused by Rickettsiae | Upper respiratory tract infections caused by Streptococcus pneumoniae
Dengue virus
Hawaii
Pathway
Enzyme-linked immunosorbent assay
Decrease (20 %)
Approved, Investigational
27396621
DrugRepV_5630Minocycline
Antiinfectives For Systemic Use
Rocky Mountain spotted fever | Typhus fever and the typhus group | Q fever | Rickettsial pox | tick fevers caused by Rickettsiae | Upper respiratory tract infections caused by Streptococcus pneumoniae
Dengue virus
H87
Pathway
Enzyme-linked immunosorbent assay
Decrease (30 %)
Approved, Investigational
27396621
DrugRepV_5631Minocycline
Antiinfectives For Systemic Use
Rocky Mountain spotted fever | Typhus fever and the typhus group | Q fever | Rickettsial pox | tick fevers caused by Rickettsiae | Upper respiratory tract infections caused by Streptococcus pneumoniae
Dengue virus
H241
Pathway
Enzyme-linked immunosorbent assay
Decrease (30 %)
Approved, Investigational
27396621
DrugRepV_5632Minocycline
Antiinfectives For Systemic Use
Rocky Mountain spotted fever | Typhus fever and the typhus group | Q fever | Rickettsial pox | tick fevers caused by Rickettsiae | Upper respiratory tract infections caused by Streptococcus pneumoniae
Dengue virus
16681
Pathway
Real-time PCR
Decrease (50 %)
Approved, Investigational
27396621
DrugRepV_5633Minocycline
Antiinfectives For Systemic Use
Rocky Mountain spotted fever | Typhus fever and the typhus group | Q fever | Rickettsial pox | tick fevers caused by Rickettsiae | Upper respiratory tract infections caused by Streptococcus pneumoniae
Dengue virus
16681
Pathway
Focus forming assay
Decrease (1 Log10 (FFU/ml))
Approved, Investigational
27396621
DrugRepV_5634Lomefloxacin
Antiinfectives For Systemic Use
Bacterial infections (respiratory tract (chronic bronchitis) and urinary tract)
Dengue virus
16681
Pathway
Enzyme-linked immunosorbent assay
No significant effect (5 %)
Approved, Investigational
27396621
DrugRepV_5635Netilmicin
Antiinfectives For Systemic Use
Bacteremia | Septicaemia | Respiratory tract infections | Skin and soft-tissue infection | Burns | Wounds | Peri-operative infections caused by susceptible strains
Dengue virus
16681
Pathway
Enzyme-linked immunosorbent assay
No significant effect (0 %)
Approved, Investigational
27396621
DrugRepV_5713Ribavirin
Antiinfectives For Systemic Use
Hepatitis C virus
Dengue virus
New Guinea C
Pathway
Fluorescence-based assay
Decrease (50 %)
Approved
20973722
DrugRepV_5723Acetylspiramycin
Antiinfectives For Systemic Use
Microbial infections
Dengue virus
New Guinea C
Pathway
Fluorescence-based assay
Decrease (50 %)
NA
20973722
DrugRepV_5743Telaprevir
Antiinfectives For Systemic Use
Hepatitis C virus
Dengue virus
DV2-NGC
Pathway
Plaque assay
Decrease (50 %)
Approved
29297305
DrugRepV_5744Asunaprevir
Antiinfectives For Systemic Use
Hepatitis C virus
Dengue virus
DV2-NGC
Pathway
Plaque assay
Decrease (50 %)
Phase III
29297305
DrugRepV_5745Boceprevir
Antiinfectives For Systemic Use
Hepatitis C virus
Dengue virus
DV2-NGC
Pathway
Real-time PCR
No significant effect
Phase II
29297305
DrugRepV_5746Telaprevir
Antiinfectives For Systemic Use
Hepatitis C virus
Dengue virus
DV2-NGC
Pathway
Real-time PCR
Decrease (2 Logs)
Approved
29297305
DrugRepV_5747Asunaprevir
Antiinfectives For Systemic Use
Hepatitis C virus
Dengue virus
DV2-NGC
Pathway
Real-time PCR
Decrease (5 Logs)
Phase III
29297305
DrugRepV_5752Nelfinavir Mesylate
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Dengue virus
DENV-2 replicon
Pathway
Luciferase reporter assay
No significant effect (0 %)
NA
28814523
DrugRepV_5779Clarithromycin
Antiinfectives For Systemic Use
NA
Dengue virus
Singapore isolates
Pathway
Plaque assay
Decrease (72 %)
NA
25251726
DrugRepV_6128Ribavirin
Antiinfectives For Systemic Use
Hepatitis C virus
Dengue virus
New Guinea C
Pathway
NA
Decrease (50 %)
Approved
29890736
DrugRepV_6138Ribavirin
Antiinfectives For Systemic Use
Hepatitis C virus
Dengue virus
New Guinea C
Pathway
DENV replicon assay
Decrease (50 %)
Approved
29672522
DrugRepV_6159Ribavirin
Antiinfectives For Systemic Use
Hepatitis C virus
Dengue virus
16681
Pathway
MTT assay
Decrease (50 %)
Approved
22068705
DrugRepV_6168Ribavirin
Antiinfectives For Systemic Use
Hepatitis C virus
Dengue virus
02--20
Pathway
Luciferase assay
Decrease (50 %)
Approved
24858611
DrugRepV_6178Ribavirin
Antiinfectives For Systemic Use
Hepatitis C virus
Dengue virus
ThNH-7/93
Pathway
Fluorescent focus-forming assay
Decrease (50 %)
Approved
22784856
DrugRepV_6182Ribavirin
Antiinfectives For Systemic Use
Hepatitis C virus
Dengue virus
New Guinea C (NGC)
Pathway
Cell proliferation assay
Decrease (50 %)
Approved
17662475
DrugRepV_6215Tetracycline
Antiinfectives For Systemic Use
Bacterial infections (Rocky Mountain spotted fever | Typhus fever | Tick fevers | Q fever | Rickettsialpox | Brill-Zinsser disease)
Dengue virus
NA
Pathway
Virus inhibition assay
Decrease (23.6 ± 2.1 %)
Approved
24522138
DrugRepV_6216Oxytetracycline
Antiinfectives For Systemic Use
Bacterial infections
Dengue virus
NA
Pathway
Virus inhibition assay
Decrease (18.8 ± 2.1 %)
Approved, Investigational, Vet approved
24522138
DrugRepV_6217Doxycycline
Antiinfectives For Systemic Use
Bacterial infections
Dengue virus
NA
Pathway
Virus inhibition assay
Decrease (50 %)
Approved
24522138
DrugRepV_6218Rolitetracycline
Antiinfectives For Systemic Use
Bacterial infection
Dengue virus
NA
Pathway
Virus inhibition assay
Decrease (32.8 ± 2.6 %)
Approved
24522138
DrugRepV_6219Ribavirin
Antiinfectives For Systemic Use
Hepatitis C virus
Dengue virus
NA
Pathway
Virus inhibition assay
Decrease (50 %)
Approved
24522138
DrugRepV_6226Ribavirin
Antiinfectives For Systemic Use
Hepatitis C virus
Dengue virus
16681
Pathway
Plaque assay
Decrease (1.75 * 105 pfu/ml)
Approved
7201778
DrugRepV_6348Ribavirin
Antiinfectives For Systemic Use
Hepatitis C virus
Dengue virus
New Guinea C (NGC)
Pathway
NA
Decrease (50 %)
Approved
26856827
DrugRepV_6491Lamivudine
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome | Hepatitis B virus
Human immunodeficiency virus
NA
Pathway
Modelling based approach
Decrease (50 %)
Approved
26796142
DrugRepV_6492Emtricitabine
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
NA
Pathway
Modelling based approach
Decrease (50 %)
Approved
26796142
DrugRepV_6493Tenofovir disoproxil Fumarate
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
NA
Pathway
Modelling based approach
Decrease (50 %)
NA
26796142
DrugRepV_6501Minocycline
Antiinfectives For Systemic Use
Rocky Mountain spotted fever | Typhus fever and the typhus group | Q fever | Rickettsial pox | tick fevers caused by Rickettsiae | Upper respiratory tract infections caused by Streptococcus pneumoniae
Human immunodeficiency virus
HIV-1ADA
Pathway
Enzyme-linked immunosorbent assay
Decrease (50 %)
Approved, Investigational
15385252
DrugRepV_6502Minocycline
Antiinfectives For Systemic Use
Rocky Mountain spotted fever | Typhus fever and the typhus group | Q fever | Rickettsial pox | tick fevers caused by Rickettsiae | Upper respiratory tract infections caused by Streptococcus pneumoniae
Human immunodeficiency virus
HIV-1ADA
Pathway
Enzyme-linked immunosorbent assay
Decrease (71-96 %)
Approved, Investigational
15385252
DrugRepV_6503Minocycline
Antiinfectives For Systemic Use
Rocky Mountain spotted fever | Typhus fever and the typhus group | Q fever | Rickettsial pox | tick fevers caused by Rickettsiae | Upper respiratory tract infections caused by Streptococcus pneumoniae
Human immunodeficiency virus
HIV-1ADA
Pathway
Enzyme-linked immunosorbent assay
Decrease (85 %)
Approved, Investigational
15385252
DrugRepV_6504Minocycline
Antiinfectives For Systemic Use
Rocky Mountain spotted fever | Typhus fever and the typhus group | Q fever | Rickettsial pox | tick fevers caused by Rickettsiae | Upper respiratory tract infections caused by Streptococcus pneumoniae
Human immunodeficiency virus
HIV-1BaL
Pathway
Enzyme-linked immunosorbent assay
Decrease (65 %)
Approved, Investigational
15385252
DrugRepV_6505Minocycline
Antiinfectives For Systemic Use
Rocky Mountain spotted fever | Typhus fever and the typhus group | Q fever | Rickettsial pox | tick fevers caused by Rickettsiae | Upper respiratory tract infections caused by Streptococcus pneumoniae
Human immunodeficiency virus
HIV-189.6
Pathway
Enzyme-linked immunosorbent assay
Decrease (NA %)
Approved, Investigational
15385252
DrugRepV_6506Minocycline
Antiinfectives For Systemic Use
Rocky Mountain spotted fever | Typhus fever and the typhus group | Q fever | Rickettsial pox | tick fevers caused by Rickettsiae | Upper respiratory tract infections caused by Streptococcus pneumoniae
Human immunodeficiency virus
HIV-1JR-FL env
Pathway
Luciferase reporter assay
Decrease (80 %)
Approved, Investigational
15385252
DrugRepV_6507Minocycline
Antiinfectives For Systemic Use
Rocky Mountain spotted fever | Typhus fever and the typhus group | Q fever | Rickettsial pox | tick fevers caused by Rickettsiae | Upper respiratory tract infections caused by Streptococcus pneumoniae
Human immunodeficiency virus
HIV-1 VSV-G env
Pathway
Luciferase reporter assay
Decrease (60 %)
Approved, Investigational
15385252
DrugRepV_6508Minocycline
Antiinfectives For Systemic Use
Rocky Mountain spotted fever | Typhus fever and the typhus group | Q fever | Rickettsial pox | tick fevers caused by Rickettsiae | Upper respiratory tract infections caused by Streptococcus pneumoniae
Human immunodeficiency virus
HIV-1 AML-V env
Pathway
Luciferase reporter assay
No significant effect (40 %)
Approved, Investigational
15385252
DrugRepV_6509Minocycline
Antiinfectives For Systemic Use
Rocky Mountain spotted fever | Typhus fever and the typhus group | Q fever | Rickettsial pox | tick fevers caused by Rickettsiae | Upper respiratory tract infections caused by Streptococcus pneumoniae
Human immunodeficiency virus
HIV-1 VSV-G env
Pathway
Luciferase reporter assay
Decrease (50 %)
Approved, Investigational
15385252
DrugRepV_6511Efavirenz
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
Wild type
Pathway
ECL RT biochemical assay
Decrease (50 %)
NA
24379202
DrugRepV_6512Etravirine
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
Wild type
Pathway
ECL RT biochemical assay
Decrease (50 %)
NA
24379202
DrugRepV_6513Rilpivirine
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
Wild type
Pathway
ECL RT biochemical assay
Decrease (50 %)
Approved
24379202
DrugRepV_6515Efavirenz
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
K103N
Pathway
ECL RT biochemical assay
Decrease (50 %)
NA
24379202
DrugRepV_6516Etravirine
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
K103N
Pathway
ECL RT biochemical assay
Decrease (50 %)
NA
24379202
DrugRepV_6517Rilpivirine
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
K103N
Pathway
ECL RT biochemical assay
Decrease (50 %)
Approved
24379202
DrugRepV_6519Efavirenz
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
Y181C
Pathway
ECL RT biochemical assay
Decrease (50 %)
NA
24379202
DrugRepV_6520Etravirine
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
Y181C
Pathway
ECL RT biochemical assay
Decrease (50 %)
NA
24379202
DrugRepV_6521Rilpivirine
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
Y181C
Pathway
ECL RT biochemical assay
Decrease (50 %)
Approved
24379202
DrugRepV_6523Efavirenz
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
Wild type
Pathway
HIV multiple-cycle replication assay
Decrease (95 %)
NA
24379202
DrugRepV_6524Etravirine
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
Wild type
Pathway
HIV multiple-cycle replication assay
Decrease (95 %)
NA
24379202
DrugRepV_6525Rilpivirine
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
Wild type
Pathway
HIV multiple-cycle replication assay
Decrease (95 %)
Approved
24379202
DrugRepV_6527Efavirenz
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
K103N
Pathway
HIV multiple-cycle replication assay
Decrease (95 %)
NA
24379202
DrugRepV_6528Etravirine
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
K103N
Pathway
HIV multiple-cycle replication assay
Decrease (95 %)
NA
24379202
DrugRepV_6529Rilpivirine
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
K103N
Pathway
HIV multiple-cycle replication assay
Decrease (95 %)
Approved
24379202
DrugRepV_6531Efavirenz
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
Y181C
Pathway
HIV multiple-cycle replication assay
Decrease (95 %)
NA
24379202
DrugRepV_6532Etravirine
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
Y181C
Pathway
HIV multiple-cycle replication assay
Decrease (95 %)
NA
24379202
DrugRepV_6533Rilpivirine
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
Y181C
Pathway
HIV multiple-cycle replication assay
Decrease (95 %)
Approved
24379202
DrugRepV_6535Efavirenz
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
K103N/Y181C
Pathway
HIV multiple-cycle replication assay
Decrease (95 %)
NA
24379202
DrugRepV_6536Etravirine
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
K103N/Y181C
Pathway
HIV multiple-cycle replication assay
Decrease (95 %)
NA
24379202
DrugRepV_6537Rilpivirine
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
K103N/Y181C
Pathway
HIV multiple-cycle replication assay
Decrease (95 %)
Approved
24379202
DrugRepV_6568Saquinavir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
HIV-1ERS104pre
Pathway
p24 assay
Decrease (50 %)
Approved, Investigational
20810732
DrugRepV_6569Amprenavir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
HIV-1ERS104pre
Pathway
p24 assay
Decrease (50 %)
Approved
20810732
DrugRepV_6570Indinavir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
HIV-1ERS104pre
Pathway
p24 assay
Decrease (50 %)
Approved
20810732
DrugRepV_6571Nelfinavir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
HIV-1ERS104pre
Pathway
p24 assay
Decrease (50 %)
Approved
20810732
DrugRepV_6572Ritonavir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
HIV-1ERS104pre
Pathway
p24 assay
Decrease (50 %)
Approved, Investigational
20810732
DrugRepV_6573Lopinavir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
HIV-1ERS104pre
Pathway
p24 assay
Decrease (50 %)
Approved
20810732
DrugRepV_6574Atazanavir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
HIV-1ERS104pre
Pathway
p24 assay
Decrease (50 %)
Approved
20810732
DrugRepV_6575Tipranavir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
HIV-1ERS104pre
Pathway
p24 assay
Decrease (50 %)
Approved, Investigational
20810732
DrugRepV_6576Darunavir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
HIV-1ERS104pre
Pathway
p24 assay
Decrease (50 %)
Approved
20810732
DrugRepV_6577Raltegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
WT
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6578Raltegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
Y143R (RAL)
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6579Raltegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
N155H(RAL)
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6580Raltegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
G140S/Q148H (RAL)
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6581Raltegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
T661(EVG)
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6582Raltegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
E92Q (EVG)
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6583Raltegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
H51Y (DTG)
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6584Raltegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
G118R (DTG)
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6585Raltegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
R263K (DTG)
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6586Raltegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
H51Y/R263K (DTG)
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6587Raltegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
E138K/R263K (DTG)
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6588Elvitegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
WT
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6589Elvitegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
Y143R (RAL)
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6590Elvitegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
N155H(RAL)
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6591Elvitegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
G140S/Q148H (RAL)
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6592Elvitegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
T661(EVG)
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6593Elvitegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
E92Q (EVG)
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6594Elvitegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
H51Y (DTG)
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6595Elvitegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
G118R (DTG)
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6596Elvitegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
R263K (DTG)
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6597Elvitegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
H51Y/R263K (DTG)
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6598Elvitegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
E138K/R263K (DTG)
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6599Dolutegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
WT
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6600Dolutegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
Y143R (RAL)
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6601Dolutegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
N155H(RAL)
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6602Dolutegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
G140S/Q148H (RAL)
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6603Dolutegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
T661(EVG)
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6604Dolutegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
E92Q (EVG)
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6605Dolutegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
H51Y (DTG)
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6606Dolutegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
G118R (DTG)
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6607Dolutegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
R263K (DTG)
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6608Dolutegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
H51Y/R263K (DTG)
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6609Dolutegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
E138K/R263K (DTG)
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6621Bictegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
WT
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6622Bictegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
Y143R (RAL)
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6623Bictegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
N155H(RAL)
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6624Bictegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
G140S/Q148H (RAL)
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6625Bictegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
T661(EVG)
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6626Bictegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
E92Q (EVG)
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6627Bictegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
H51Y (DTG)
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6628Bictegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
G118R (DTG)
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6629Bictegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
R263K (DTG)
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6630Bictegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
H51Y/R263K (DTG)
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6631Bictegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
E138K/R263K (DTG)
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6632Raltegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
M50I
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6633Raltegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
L74M
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6634Raltegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
T97A
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6635Raltegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
S119R
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6636Raltegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
E138K
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6637Raltegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
G140S
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6638Raltegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
Q146L
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6639Raltegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
Q146P
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6640Raltegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
Q148H
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6641Raltegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
Q148K
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6642Raltegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
Q148R
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6643Raltegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
S153Y
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6644Elvitegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
M50I
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6645Elvitegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
L74M
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6646Elvitegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
T97A
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6647Elvitegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
S119R
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6648Elvitegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
E138K
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6649Elvitegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
G140S
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6650Elvitegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
Q146L
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6651Elvitegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
Q146P
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6652Elvitegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
Q148H
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6653Elvitegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
Q148K
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6654Elvitegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
Q148R
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6655Elvitegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
S153Y
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6656Dolutegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
M50I
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6657Dolutegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
L74M
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6658Dolutegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
T97A
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6659Dolutegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
S119R
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6660Dolutegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
E138K
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6661Dolutegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
G140S
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6662Dolutegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
Q146L
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6663Dolutegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
Q146P
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6664Dolutegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
Q148H
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6665Dolutegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
Q148K
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6666Dolutegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
Q148R
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6667Dolutegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
S153Y
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6680Bictegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
M50I
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6681Bictegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
L74M
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6682Bictegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
T97A
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6683Bictegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
S119R
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6684Bictegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
E138K
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6685Bictegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
G140S
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6686Bictegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
Q146L
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6687Bictegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
Q146P
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6688Bictegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
Q148H
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6689Bictegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
Q148K
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6690Bictegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
Q148R
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6691Bictegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
S153Y
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6692Raltegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
G140A/Q148H
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6693Raltegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
Y143R/Q148H
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6694Raltegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
Q148H/N155H
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6695Raltegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
E138K/Q148K
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6696Raltegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
G140A/Q148K
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6697Raltegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
G140S/Q148K
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6698Raltegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
E138A/Q148R
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6699Raltegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
E138K/Q148R
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6700Raltegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
G140A/Q148R
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6701Raltegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
G140C/Q148R
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6702Raltegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
G140S/Q148R
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6703Raltegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
Q148R/N155H
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6704Elvitegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
G140A/Q148H
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6705Elvitegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
Y143R/Q148H
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6706Elvitegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
Q148H/N155H
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6707Elvitegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
E138K/Q148K
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6708Elvitegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
G140A/Q148K
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6709Elvitegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
G140S/Q148K
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6710Elvitegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
E138A/Q148R
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6711Elvitegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
E138K/Q148R
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6712Elvitegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
G140A/Q148R
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6713Elvitegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
G140C/Q148R
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6714Elvitegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
G140S/Q148R
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6715Elvitegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
Q148R/N155H
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6716Dolutegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
G140A/Q148H
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6717Dolutegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
Y143R/Q148H
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6718Dolutegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
Q148H/N155H
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6719Dolutegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
E138K/Q148K
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6720Dolutegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
G140A/Q148K
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6721Dolutegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
G140S/Q148K
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6722Dolutegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
E138A/Q148R
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6723Dolutegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
E138K/Q148R
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6724Dolutegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
G140A/Q148R
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6725Dolutegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
G140C/Q148R
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6726Dolutegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
G140S/Q148R
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6727Dolutegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
Q148R/N155H
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6740Bictegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
G140A/Q148H
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6741Bictegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
Y143R/Q148H
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6742Bictegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
Q148H/N155H
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6743Bictegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
E138K/Q148K
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6744Bictegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
G140A/Q148K
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6745Bictegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
G140S/Q148K
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6746Bictegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
E138A/Q148R
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6747Bictegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
E138K/Q148R
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6748Bictegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
G140A/Q148R
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6749Bictegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
G140C/Q148R
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6750Bictegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
G140S/Q148R
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6751Bictegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
Q148R/N155H
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6752Raltegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
T66I/E157Q
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6753Raltegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
E92Q/N155H
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6754Raltegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
G140S/N155H
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6755Raltegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
Y143H/N155H
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6756Raltegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
Y143R/N155H
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6757Raltegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
N155H/G163R
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6758Elvitegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
T66I/E157Q
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6759Elvitegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
E92Q/N155H
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6760Elvitegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
G140S/N155H
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6761Elvitegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
Y143H/N155H
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6762Elvitegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
Y143R/N155H
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6763Elvitegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
N155H/G163R
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6764Dolutegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
T66I/E157Q
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6765Dolutegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
E92Q/N155H
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6766Dolutegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
G140S/N155H
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6767Dolutegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
Y143H/N155H
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6768Dolutegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
Y143R/N155H
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6769Dolutegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
N155H/G163R
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6776Bictegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
T66I/E157Q
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6777Bictegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
E92Q/N155H
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6778Bictegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
G140S/N155H
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6779Bictegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
Y143H/N155H
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6780Bictegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
Y143R/N155H
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6781Bictegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
N155H/G163R
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6782Raltegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
97A/Y143R/Q148H
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6783Raltegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
T97A/Q148H/N155H
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6784Raltegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
E138K/G140A/Q148K
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6785Raltegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
L74M/G140A/Q148R
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6786Raltegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
L74M/G140C/Q148R
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6787Raltegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
E138K/G140C/Q148R
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6788Raltegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
E138A/S147G/Q148R
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6789Elvitegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
97A/Y143R/Q148H
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6790Elvitegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
T97A/Q148H/N155H
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6791Elvitegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
E138K/G140A/Q148K
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6792Elvitegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
L74M/G140A/Q148R
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6793Elvitegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
L74M/G140C/Q148R
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6794Elvitegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
E138K/G140C/Q148R
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6795Elvitegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
E138A/S147G/Q148R
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6796Dolutegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
97A/Y143R/Q148H
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6797Dolutegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
T97A/Q148H/N155H
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6798Dolutegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
E138K/G140A/Q148K
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6799Dolutegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
L74M/G140A/Q148R
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6800Dolutegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
L74M/G140C/Q148R
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6801Dolutegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
E138K/G140C/Q148R
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6802Dolutegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
E138A/S147G/Q148R
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6810Bictegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
97A/Y143R/Q148H
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6811Bictegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
T97A/Q148H/N155H
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6812Bictegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
E138K/G140A/Q148K
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6813Bictegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
L74M/G140A/Q148R
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6814Bictegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
L74M/G140C/Q148R
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6815Bictegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
E138K/G140C/Q148R
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6816Bictegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
E138A/S147G/Q148R
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6817Raltegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
T66I/T97A/E157Q
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6818Raltegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
T97A/Y143R/N155H
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6819Raltegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
G140S/Y143R/N155H
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6820Raltegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
E92Q/N155H/G163R
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6821Elvitegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
T66I/T97A/E157Q
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6822Elvitegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
T97A/Y143R/N155H
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6823Elvitegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
G140S/Y143R/N155H
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6824Elvitegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
E92Q/N155H/G163R
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6825Dolutegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
T66I/T97A/E157Q
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6826Dolutegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
T97A/Y143R/N155H
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6827Dolutegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
G140S/Y143R/N155H
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6828Dolutegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
E92Q/N155H/G163R
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6833Bictegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
T66I/T97A/E157Q
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6834Bictegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
T97A/Y143R/N155H
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6835Bictegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
G140S/Y143R/N155H
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6836Bictegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
E92Q/N155H/G163R
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6837Raltegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
T97A/G140S/Q148H
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6838Raltegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
E138A/G140S/Q148H
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6839Raltegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
E138K/G140S/Q148H
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6840Raltegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
G140S/Y143R/Q148H
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6841Raltegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
G140S/Q148H/N155H
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6842Raltegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
G140S/Q148H/G163K
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6843Elvitegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
T97A/G140S/Q148H
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6844Elvitegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
E138A/G140S/Q148H
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6845Elvitegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
E138K/G140S/Q148H
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6846Elvitegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
G140S/Y143R/Q148H
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6847Elvitegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
G140S/Q148H/N155H
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6848Elvitegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
G140S/Q148H/G163K
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6849Dolutegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
T97A/G140S/Q148H
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6850Dolutegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
E138A/G140S/Q148H
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6851Dolutegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
E138K/G140S/Q148H
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6852Dolutegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
G140S/Y143R/Q148H
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6853Dolutegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
G140S/Q148H/N155H
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6854Dolutegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
G140S/Q148H/G163K
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6861Bictegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
T97A/G140S/Q148H
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6862Bictegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
E138A/G140S/Q148H
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6863Bictegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
E138K/G140S/Q148H
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6864Bictegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
G140S/Y143R/Q148H
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6865Bictegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
G140S/Q148H/N155H
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6866Bictegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
G140S/Q148H/G163K
Pathway
Single-round viral replication assay
Decrease (50 %)
Approved
29769116
DrugRepV_6926AzidoThymidine
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
IIIB
Pathway
MTT assay
Decrease (50 %)
Approved
25970561
DrugRepV_6956AzidoThymidine
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
ROD
Pathway
MTT assay
Decrease (50 %)
Approved
25970561
DrugRepV_6958Ribavirin
Antiinfectives For Systemic Use
Hepatitis C virus
Human immunodeficiency virus
NA
Pathway
NA
Decrease (50 %)
Approved
15200845
DrugRepV_6959Lamivudine
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome | Hepatitis B virus
Human immunodeficiency virus
NA
Pathway
NA
Decrease (50 %)
Approved
15200845
DrugRepV_6960Zidovudine
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome/AIDS
Human immunodeficiency virus
NA
Pathway
NA
Decrease (50 %)
Approved
15200845
DrugRepV_6961Saquinavir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
NA
Pathway
NA
Decrease (50 %)
Approved, Investigational
15200845
DrugRepV_6962Nelfinavir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
NA
Pathway
NA
Decrease (95 %)
Approved
15200845
DrugRepV_6963Indinavir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Human immunodeficiency virus
NA
Pathway
NA
Decrease (50 %)
Approved
15200845
DrugRepV_7011Nelfinavir Mesylate
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Japanese encephalitis virus
AT31
Pathway
Luciferase reporter assay
Decrease (50 %)
NA
28814523
DrugRepV_7020Nelfinavir Mesylate
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Japanese encephalitis virus
AT31
Pathway
Plaque assay
Decrease (3 Logs)
NA
28814523
DrugRepV_7025Nelfinavir Mesylate
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Japanese encephalitis virus
AT31
Pathway
Real-time PCR
Decrease (0.1 %)
NA
28814523
DrugRepV_7030Nelfinavir Mesylate
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Japanese encephalitis virus
AT31
Pathway
Immunoflourescence assay
Decrease (100 %)
NA
28814523
DrugRepV_7035Nelfinavir Mesylate
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Japanese encephalitis virus
AT31
Pathway
Luciferase reporter assay
Decrease (70 %)
NA
28814523
DrugRepV_7040Nelfinavir Mesylate
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Japanese encephalitis virus
AT31
Pathway
Luciferase reporter assay
Decrease (100 %)
NA
28814523
DrugRepV_7045Nelfinavir Mesylate
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
West Nile virus
WNV replicon
Pathway
Luciferase reporter assay
Decrease (72 %)
NA
28814523
DrugRepV_7089Teicoplanin
Antiinfectives For Systemic Use
Bacterial infections
Polio virus
Sabin
Pathway
Plaque assay
No significant effect
Approved
26585243
DrugRepV_7447Ribavirin
Antiinfectives For Systemic Use
Hepatitis C virus
West Nile virus
New York
Pathway
Visual assay
Decrease (50 %)
Approved
12076755
DrugRepV_7448Ribavirin
Antiinfectives For Systemic Use
Hepatitis C virus
West Nile virus
Uganda strain B 956
Pathway
Visual assay
Decrease (50 %)
Approved
12076755
DrugRepV_7459Ribavirin
Antiinfectives For Systemic Use
Hepatitis C virus
West Nile virus
New York
Pathway
NR assay
Decrease (50 %)
Approved
12076755
DrugRepV_7460Ribavirin
Antiinfectives For Systemic Use
Hepatitis C virus
West Nile virus
Uganda strain B 956
Pathway
NR assay
Decrease (50 %)
Approved
12076755
DrugRepV_7506Ribavirin
Antiinfectives For Systemic Use
Hepatitis C virus
West Nile virus
New York
Pathway
Visual assay
Decrease (50 %)
Approved
12076755
DrugRepV_7511Ribavirin
Antiinfectives For Systemic Use
Hepatitis C virus
West Nile virus
New York
Pathway
Virus yield reduction assay
Decrease (90 %)
Approved
12076755
DrugRepV_7519Rifampicin
Antiinfectives For Systemic Use
Tuberculosis and Tuberculosis-related mycobacterial infections
Vaccinia virus
NA
Pathway
Plaque assay
Decrease (Complete inhibition Plaque size)
Approved
4321450
DrugRepV_7525Telaprevir
Antiinfectives For Systemic Use
Hepatitis C virus
Enterovirus
US/KY/14-18953
Pathway
Cytopathic effect (CPE) assay
Decrease (50 %)
Approved
30674624
DrugRepV_7526Telaprevir
Antiinfectives For Systemic Use
Hepatitis C virus
Enterovirus
US/MO/14-18949
Pathway
Cytopathic effect (CPE) assay
Decrease (50 %)
Approved
30674624
DrugRepV_7527Telaprevir
Antiinfectives For Systemic Use
Hepatitis C virus
Enterovirus
US/MO/14-18947
Pathway
Cytopathic effect (CPE) assay
Decrease (50 %)
Approved
30674624
DrugRepV_7528Telaprevir
Antiinfectives For Systemic Use
Hepatitis C virus
Enterovirus
US/IL/14-18952
Pathway
Cytopathic effect (CPE) assay
Decrease (50 %)
Approved
30674624
DrugRepV_7529Telaprevir
Antiinfectives For Systemic Use
Hepatitis C virus
Enterovirus
US/IL/14-18956
Pathway
Cytopathic effect (CPE) assay
Decrease (50 %)
Approved
30674624
DrugRepV_7530Telaprevir
Antiinfectives For Systemic Use
Hepatitis C virus
Enterovirus
US/KY/14-18953
Pathway
Cytopathic effect (CPE) assay
Decrease (50 %)
Approved
30674624
DrugRepV_7531Telaprevir
Antiinfectives For Systemic Use
Hepatitis C virus
Enterovirus
US/KY/14-18953
Pathway
Cytopathic effect (CPE) assay
Decrease (50 %)
Approved
30674624
DrugRepV_7532Telaprevir
Antiinfectives For Systemic Use
Hepatitis C virus
Enterovirus
US/KY/14-18953
Pathway
Cytopathic effect (CPE) assay
Decrease (50 %)
Approved
30674624
DrugRepV_7533Telaprevir
Antiinfectives For Systemic Use
Hepatitis C virus
Enterovirus
US/KY/14-18953
Pathway
Cytopathic effect (CPE) assay
Decrease (50 %)
Approved
30674624
DrugRepV_7550Nelfinavir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
SARS Coronavirus-2
NA
NA
RT-PCR
Decrease (50 %)
Approved
32438446
DrugRepV_7551Nelfinavir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
SARS Coronavirus-2
NA
NA
RT-PCR
Decrease (90 %)
Approved
32438446
DrugRepV_7560Atazanavir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
SARS Coronavirus-2
Brazil/RJ-314/2020
NA
RT-PCR
Decrease (50 %)
Approved
32438446
DrugRepV_7561Atazanavir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
SARS Coronavirus-2
Brazil/RJ-314/2020
NA
RT-PCR
Decrease (90 %)
Approved
32438446
DrugRepV_7562Azithromycin
Antiinfectives For Systemic Use
Microbial infections
SARS Coronavirus-2
BavPat1
NA
RT-PCR
Decrease (50 %)
Approved
32438446
DrugRepV_7563Azithromycin
Antiinfectives For Systemic Use
Microbial infections
SARS Coronavirus-2
BavPat1
NA
RT-PCR
Decrease (90 %)
Approved
32438446
DrugRepV_7568Nelfinavir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
SARS Coronavirus-2
NA
NA
RT-PCR
Decrease (50 %)
Approved
32438446
DrugRepV_7602Lopinavir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
SARS Coronavirus-2
NA
NA
RT-PCR
Decrease (50 %)
Approved
32438446
DrugRepV_7603Lopinavir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
SARS Coronavirus-2
NA
NA
RT-PCR
Decrease (90 %)
Approved
32438446
DrugRepV_7620Umifenovir
Antiinfectives For Systemic Use
Prophylaxis/treatment of influenza in Russia and China
SARS Coronavirus-2
BavPat1
NA
RT-PCR
Decrease (50 %)
Investigational
32438446
DrugRepV_7621Umifenovir
Antiinfectives For Systemic Use
Prophylaxis/treatment of influenza in Russia and China
SARS Coronavirus-2
BavPat1
NA
RT-PCR
Decrease (90 %)
Investigational
32438446
DrugRepV_7622Anidulafungin
Antiinfectives For Systemic Use
Invasive candidiasis/candidaemia
SARS Coronavirus-2
?CoV/KOR/KCDC03/2020)
NA
Immunofluorescence
Decrease (50 %)
Approved, Investigational
32438446
DrugRepV_7623Anidulafungin
Antiinfectives For Systemic Use
Invasive candidiasis/candidaemia
SARS Coronavirus-2
?CoV/KOR/KCDC03/2020)
NA
Immunofluorescence
Decrease (90 %)
Approved, Investigational
32438446
DrugRepV_7625Lopinavir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
SARS Coronavirus-2
?CoV/KOR/KCDC03/2020
NA
Immunofluorescence
Decrease (50 %)
Approved
32438446
DrugRepV_7626Lopinavir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
SARS Coronavirus-2
?CoV/KOR/KCDC03/2020
NA
Immunofluorescence
Decrease (90 %)
Approved
32438446
DrugRepV_7629Saquinavir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
SARS Coronavirus-2
NA
NA
RT-PCR
Decrease (50 %)
Approved, Investigational
32438446
DrugRepV_7630Saquinavir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
SARS Coronavirus-2
NA
NA
RT-PCR
Decrease (90 %)
Approved, Investigational
32438446
DrugRepV_7633Ritonavir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
SARS Coronavirus-2
NA
NA
RT-PCR
Decrease (50 %)
Approved, Investigational
32438446
DrugRepV_7634Ritonavir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
SARS Coronavirus-2
NA
NA
RT-PCR
Decrease (90 %)
Approved, Investigational
32438446
DrugRepV_7635Atazanavir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
SARS Coronavirus-2
NA
NA
RT-PCR
Decrease (50 %)
Approved
32438446
DrugRepV_7636Atazanavir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
SARS Coronavirus-2
NA
NA
RT-PCR
Decrease (90 %)
Approved
32438446
DrugRepV_7643Tipranavir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
SARS Coronavirus-2
NA
NA
RT-PCR
Decrease (50 %)
Approved, Investigational
32438446
DrugRepV_7644Tipranavir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
SARS Coronavirus-2
NA
NA
RT-PCR
Decrease (90 %)
Approved, Investigational
32438446
DrugRepV_7645Dolutegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
SARS Coronavirus-2
BavPat1
NA
RT-PCR
Decrease (50 %)
Approved
32438446
DrugRepV_7646Dolutegravir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
SARS Coronavirus-2
BavPat1
NA
RT-PCR
Decrease (90 %)
Approved
32438446
DrugRepV_7647Lopinavir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
SARS Coronavirus-2
?CoV/KOR/KCDC03/2020)
NA
Cytopathic effect (CPE) assay
Decrease (50 %)
Approved
32438446
DrugRepV_7648Lopinavir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
SARS Coronavirus-2
?CoV/KOR/KCDC03/2020)
NA
Cytopathic effect (CPE) assay
Decrease (90 %)
Approved
32438446
DrugRepV_7652Amprenavir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
SARS Coronavirus-2
NA
NA
RT-PCR
Decrease (50 %)
Approved
32438446
DrugRepV_7653Amprenavir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
SARS Coronavirus-2
NA
NA
RT-PCR
Decrease (90 %)
Approved
32438446
DrugRepV_7655Penciclovir
Antiinfectives For Systemic Use
Recurrent cold sores on the lips and face from Herpesvirus invections
SARS Coronavirus-2
Wuhan/WIV04/2019
NA
qRT-PCR/ NP expression/Immunofluorescence
Decrease (50 %)
Approved
32438446
DrugRepV_7656Penciclovir
Antiinfectives For Systemic Use
Recurrent cold sores on the lips and face from Herpesvirus invections
SARS Coronavirus-2
Wuhan/WIV04/2019
NA
qRT-PCR/ NP expression/Immunofluorescence
Decrease (90 %)
Approved
32438446
DrugRepV_7657Darunavir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
SARS Coronavirus-2
NA
NA
RT-PCR
Decrease (50 %)
Approved
32438446
DrugRepV_7658Darunavir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
SARS Coronavirus-2
NA
NA
RT-PCR
Decrease (90 %)
Approved
32438446
DrugRepV_7659Ribavirin
Antiinfectives For Systemic Use
Hepatitis C virus
SARS Coronavirus-2
Wuhan/WIV04/2022
NA
qRT-PCR/ NP expression/Immunofluorescence
Decrease (50 %)
Approved
32438446
DrugRepV_7660Ribavirin
Antiinfectives For Systemic Use
Hepatitis C virus
SARS Coronavirus-2
Wuhan/WIV04/2022
NA
qRT-PCR/ NP expression/Immunofluorescence
Decrease (90 %)
Approved
32438446
DrugRepV_7661Indinavir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
SARS Coronavirus-2
NA
NA
RT-PCR
Decrease (50 %)
Approved
32438446
DrugRepV_7662Indinavir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
SARS Coronavirus-2
NA
NA
RT-PCR
Decrease (90 %)
Approved
32438446
DrugRepV_7680Clofazamine
Antiinfectives For Systemic Use
Lepromatous leprosy
SARS Coronavirus-2
NA
NA
NA
Decrease (50 %)
Approved
32577649
DrugRepV_7682Entecavir
Antiinfectives For Systemic Use
Hepatitis B virus
SARS Coronavirus-2
NA
NA
Decrease (50 %)
Approved
32577649
DrugRepV_7708Lopinavir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
SARS Coronavirus-2
NA
Plaque reduction assay
Decrease (50 %)
Approved
32532085
DrugRepV_7712Clofazimine
Antiinfectives For Systemic Use
Lepromatous leprosy
SARS Coronavirus-2
SARS-CoV-2-USA-WA1/2020
NA
Immunofluorescence
Decrease (50 %)
Approved
32707573
DrugRepV_7726Clofazimine
Antiinfectives For Systemic Use
Lepromatous leprosy
SARS Coronavirus-2
SARS-CoV-2-USA-WA1/2020
NA
Immunofluorescence
Decrease (50 %)
Approved
32707573
DrugRepV_7754Clofazimine
Antiinfectives For Systemic Use
Lepromatous leprosy
SARS Coronavirus-2
SARS-CoV-2-USA-WA1/2020
NA
Immunofluorescence
Decrease (50 %)
Approved
32707573
DrugRepV_7774Ritonavir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
SARS Coronavirus-2
NA
NA
NA
Decrease (50 %)
Approved, Investigational
32687696
DrugRepV_8144Idoxuridine
Antiinfectives For Systemic Use
Keratoconjunctivitis and Keratitis caused by herpes simplex virus
Vaccinia virus
NA
Pathway
NA
Decrease (85.8 %)
Approved, Investigational
32708182
DrugRepV_8167Adefovir dipivoxil
Antiinfectives For Systemic Use
Hepatitis B virus
Vaccinia virus
NA
Pathway
NA
Decrease (99.8 %)
Approved
32708182
DrugRepV_8193AT13387
Antiinfectives For Systemic Use
Hepatitis C virus
Vaccinia virus
NA
Pathway
NA
Decrease (99.8 %)
Phase III
32708182
DrugRepV_8277Asunaprevir
Antiinfectives For Systemic Use
Hepatitis C virus
Zika virus
NA
NA
MTT assay
Decrease (50 %)
Phase III
32488021
DrugRepV_8278Simeprevir
Antiinfectives For Systemic Use
Hepatitis C virus
Zika virus
NA
NA
MTT assay
Decrease (50 %)
Approved
32488021
DrugRepV_8299Efavirenz
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Zika virus
Paraiba_01
NA
Plaque assay
Decrease (50 %)
NA
32326119
DrugRepV_8300Efavirenz
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Zika virus
MR-766
NA
Plaque assay
Decrease (50 %)
NA
32326119
DrugRepV_8301Efavirenz
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
West Nile virus
Eg101
Pathway
Plaque assay
Decrease (50 %)
NA
32326119
DrugRepV_8302Efavirenz
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
West Nile virus
13-104
Pathway
Plaque assay
Decrease (50 %)
NA
32326119
DrugRepV_8303Tipranavir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Zika virus
Paraiba_01
NA
Plaque assay
Decrease (50 %)
Approved, Investigational
32326119
DrugRepV_8304Tipranavir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
Zika virus
MR-766
NA
Plaque assay
Decrease (50 %)
Approved, Investigational
32326119
DrugRepV_8305Tipranavir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
West Nile virus
Eg101
Pathway
Plaque assay
Decrease (50 %)
Approved, Investigational
32326119
DrugRepV_8306Tipranavir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
West Nile virus
13-104
Pathway
Plaque assay
Decrease (50 %)
Approved, Investigational
32326119
DrugRepV_8307Dasabuvir
Antiinfectives For Systemic Use
Hepatitis C virus
Zika virus
Paraiba_01
NA
Plaque assay
Decrease (50 %)
Approved
32326119
DrugRepV_8308Dasabuvir
Antiinfectives For Systemic Use
Hepatitis C virus
Zika virus
MR-766
NA
Plaque assay
Decrease (50 %)
Approved
32326119
DrugRepV_8309Dasabuvir
Antiinfectives For Systemic Use
Hepatitis C virus
West Nile virus
Eg101
Pathway
Plaque assay
Decrease (50 %)
Approved
32326119
DrugRepV_8310Dasabuvir
Antiinfectives For Systemic Use
Hepatitis C virus
West Nile virus
13-104
Pathway
Plaque assay
Decrease (50 %)
Approved
32326119
DrugRepV_8326Tenofovir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
SARS Coronavirus-2
Experimental
NA
Cytopathic effect (CPE) assay
Decrease (50 %)
Approved, Investigational
32429580
DrugRepV_8330Lamivudine
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome | Hepatitis B virus
SARS Coronavirus-2
Experimental
NA
Cytopathic effect (CPE) assay
Decrease (50 %)
Approved
32429580
DrugRepV_8332Emtricitabine
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
SARS Coronavirus-2
Experimental
NA
Cytopathic effect (CPE) assay
Decrease (50 %)
Approved
32429580
DrugRepV_8338Nelfinavir
Antiinfectives For Systemic Use
Acquired immunodeficiency syndrome
SARS Coronavirus-2
NA
NA
NA
Decrease (100 %)
Approved
32374457
DrugRepV_8451Sofosbuvir
Antiinfectives For Systemic Use
Hepatitis C virus | Acquired immunodeficiency syndrome
Yellow fever virus
YFV17D
Pathway
NA
Decrease (50 %)
Approved
30699122
DrugRepV_8452Itraconazole
Antiinfectives For Systemic Use
Fungal infections (Pulmonary and extrapulmonary blastomycosis, Histoplasmosis, Aspergillosis, and Onychomycosis)
Influenza virus
PR8M
Pathway
MTT assay
Decrease (50 %)
Approved, Investigational
30866762
DrugRepV_8453Itraconazole
Antiinfectives For Systemic Use
Fungal infections (Pulmonary and extrapulmonary blastomycosis, Histoplasmosis, Aspergillosis, and Onychomycosis)
Influenza virus
PR8M
Pathway
MTT assay
Decrease (90 %)
Approved, Investigational
30866762
DrugRepV_8454Posaconazole
Antiinfectives For Systemic Use
Fungal infections (Aspergillus and Candida infections)
Influenza virus
PR8M
Pathway
MTT assay
Decrease (50 %)
Approved, Investigational, Vet approved
30866762
DrugRepV_8455Posaconazole
Antiinfectives For Systemic Use
Fungal infections (Aspergillus and Candida infections)
Influenza virus
PR8M
Pathway
MTT assay
Decrease (90 %)
Approved, Investigational, Vet approved
30866762